SCHEMBL6204081

SCHEMBL6204081

O=C(c1ccccc1)C(Cc1ccc(Cl)cc1Cl)c1cccnn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.42
CYP3A4 P08684 1/20 0.42
PDPK1 O15530 1/20 0.41
HDAC8 Q9BY41 8/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NR4A1 P22736 1/20 0.39
NR4A2 P43354 1/20 0.39
NR4A3 Q92570 1/20 0.39
TSHR P16473 1/20 0.39
MAPT P10636 1/20 0.38
EPHX1 P07099 2/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
ATM Q13315 1/20 0.38
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204074 0.83 MDM2 (0.41) TSHR
SCHEMBL6400617 0.75 NPC1 (0.44) MAPTL3MBTL1CYP1A2
SCHEMBL29926553 0.74 PDPK1 (0.53) PDPK1HDAC8HDAC3HDAC1HDAC2
SCHEMBL10829635 0.74 PDPK1 (0.53) PDPK1HDAC8HDAC3HDAC1HDAC2
SCHEMBL6005346 0.70 HDAC8 (0.54) CYP2C9CYP3A4PDPK1HDAC8HDAC3
SCHEMBL6202771 0.67 KMT2A (0.54) PDPK1HDAC8HDAC3HDAC1HDAC2
SCHEMBL11851540 0.66 HDAC8 (0.44) CYP2C9CYP3A4PDPK1HDAC8HDAC3
SCHEMBL3371893 0.66 FFAR2 (0.42) TSHRL3MBTL1MEN1CYP1A2KMT2A
SCHEMBL11458388 0.66 IDO1 (0.49) CYP2C9CYP3A4HDAC8HDAC3HDAC1
SCHEMBL11857052 0.65 HDAC8 (0.55) CYP2C9CYP3A4HDAC8HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed