SCHEMBL6204074

SCHEMBL6204074

O=C(c1ccccc1)C(Cc1ccc(Cl)cc1)c1cccnn1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 2/20 0.41
PTPN1 P18031 11/20 0.40
EP300 Q09472 1/20 0.38
TSHR P16473 1/20 0.38
FFAR2 O15552 1/20 0.38
NTSR1 P30989 1/20 0.38
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6400617 0.90 NPC1 (0.44) MDM2PTPN1EP300
SCHEMBL6204081 0.83 CYP2C9 (0.42) TSHR
SCHEMBL3371893 0.83 FFAR2 (0.42) EP300TSHRFFAR2PPARGPPARA
SCHEMBL6203529 0.74 TSHR (0.52) PTPN1TSHR
SCHEMBL11307784 0.73 MDM2 (0.51) MDM2PPARGPPARA
SCHEMBL6204077 0.73 MGAM (0.50) TSHRFFAR2
SCHEMBL6201491 0.72 TSHR (0.50) TSHR
SCHEMBL6203634 0.72 NTSR1 (0.57) MDM2PTPN1NTSR1PPARGPPARA
SCHEMBL1127590 0.71 KMT2A (0.46) TSHRPPARGPPARA
SCHEMBL10988389 0.71 MDM2 (0.53) MDM2PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed