SCHEMBL6203495

SCHEMBL6203495

CCCN(CO)c1nc(NCc2c(O)cc(OC)cc2O)c2[nH]nnc2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRUNE1 Q86TP1 1/20 0.35
PDE5A O76074 2/20 0.33
PDE4D Q08499 2/20 0.33
PDE6C P51160 1/20 0.33
CCNE2 O96020 2/20 0.31
CCNE1 P24864 2/20 0.31
CDK2 P24941 2/20 0.31
CCNT1 O60563 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK7 P50613 1/20 0.31
CDK9 P50750 1/20 0.31
CCNH P51946 1/20 0.31
MNAT1 P51948 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
PDE10A Q9Y233 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203494 0.86 PRUNE1 (0.40) PRUNE1PDE5APDE4DPDE6CCCNE2
SCHEMBL6205414 0.83 HMGCR (0.32) PRUNE1
SCHEMBL6204811 0.80 PRUNE1 (0.32) PRUNE1PDE5APDE4DPDE6CCCNE1
SCHEMBL6204719 0.79 PGK1 (0.33)
SCHEMBL6202760 0.78 CDK1 (0.40) PRUNE1PDE4DCCNE2CCNE1CDK2
SCHEMBL3445847 0.76 CDK1 (0.39) CCNE2CCNE1CDK2CCNT1CDK1
SCHEMBL6205608 0.75 PARP1 (0.36) PRUNE1PDE5APDE4DPDE6C
SCHEMBL6203171 0.75 CCNE1 (0.37) CCNE2CCNE1CDK2CCNT1CDK7
SCHEMBL6204186 0.75 PDE5A (0.36) PRUNE1PDE5APDE4DPDE6CCCNE2
SCHEMBL3445684 0.74 CDK1 (0.39) CCNE2CCNE1CDK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed