SCHEMBL6206095

SCHEMBL6206095

COC(=O)c1cc2c3c(cc([N+](=O)[O-])c2[nH]1)N(C(=O)OC(C)(C)C)CC3CO

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.40
NR3C2 P08235 1/20 0.32
UCHL1 P09936 1/20 0.31
USP30 Q70CQ3 1/20 0.31
FBP1 P09467 7/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
NR1H2 P55055 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205393 0.80 HDAC1 (0.35) XDHHDAC1HDAC6NR1H2
SCHEMBL4590751 0.80 ADH1A (0.36) HDAC1HDAC6
SCHEMBL6205186 0.79 P4HB (0.47) XDHFBP1
SCHEMBL7954292 0.78 ADH1A (0.32) HDAC1HDAC6NR1H2
SCHEMBL3558952 0.73 ADH1A (0.47) HDAC1HDAC6
SCHEMBL5623265 0.72 P4HB (0.47) XDHFBP1
SCHEMBL6618596 0.71 ADH1A (0.46) XDH
SCHEMBL7092620 0.71 SRD5A2 (0.42)
SCHEMBL6852340 0.70 ADH1A (0.44)
SCHEMBL12596983 0.68 ADH1A (0.38) HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0938474-B1 CYCLOPROPYLINDOLE COMPOUNDS AND THEIR USE AS PRODRUGS AUCKLAND UNISERVICES LTD (NZ) 2005-11-23 EP disclosed
US-6130237-A Condensed N-aclyindoles as antitumor agents CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-10-10 US disclosed