SCHEMBL6207249

SCHEMBL6207249

C=C(N)C(=O)OC(=O)c1cccc(Cl)c1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
L3MBTL1 Q9Y468 3/20 0.42
ALOX12 P18054 1/20 0.42
ERCC5 P28715 1/20 0.41
FEN1 P39748 1/20 0.41
PKM P14618 4/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 2/20 0.40
ATM Q13315 1/20 0.40
LMNA P02545 1/20 0.40
P2RX7 Q99572 1/20 0.40
RAB9A P51151 3/20 0.38
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 2/20 0.38
JAK2 O60674 1/20 0.38
GAA P10253 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6206781 0.87 RAB9A (0.50) L3MBTL1PKMALDH1A1KDM4ELMNA
SCHEMBL5955449 0.82 TSHR (0.63) TSHRL3MBTL1ALOX12ERCC5FEN1
SCHEMBL36590 0.75 TSHR (0.63) TSHRL3MBTL1ALOX12ERCC5FEN1
SCHEMBL29566931 0.75 TSHR (0.63) TSHRL3MBTL1ALOX12ERCC5FEN1
SCHEMBL6207827 0.75 HPGD (0.52) TSHRL3MBTL1ALDH1A1KDM4ELMNA
SCHEMBL6208654 0.74 CES2 (0.50) PKMALDH1A1ATMRAB9AHPGD
SCHEMBL7578668 0.74 TSHR (0.57) TSHRL3MBTL1ALOX12ERCC5FEN1
SCHEMBL6207031 0.73 CES2 (0.47) L3MBTL1PKMALDH1A1LMNARAB9A
SCHEMBL5955453 0.73 TSHR (0.56) TSHRL3MBTL1ALOX12ERCC5FEN1
SCHEMBL6205116 0.73 NPC1 (0.50) PKMALDH1A1LMNARAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532128-A1 INHIBITORS OF HCV NS5B POLYMERASE Pharmacia & Upjohn Company LLC (US) 2005-05-25 EP disclosed
WO-2004002977-A1 INHIBITORS OF HCV NS5B POLYMERASE PHARMACIA & UPJOHN COMPANY LLC (US) 2004-01-08 WO disclosed