SCHEMBL6207258

SCHEMBL6207258

CCNCc1cccc(CNC(=O)c2c[nH]c3c(Cl)cccc3c2=O)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.51
RAB9A P51151 4/20 0.51
ADORA2A P29274 7/20 0.48
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
BACE1 P56817 2/20 0.47
NR4A2 P43354 1/20 0.46
NPC1 O15118 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
MAPK10 P53779 1/20 0.46
HSD17B10 Q99714 1/20 0.46
ADORA1 P30542 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6206360 0.94 ADORA2A (0.51) POLBRAB9AADORA2AALDH1A1MEN1
SCHEMBL6205434 0.83 POLB (0.57) POLBRAB9ABACE1NPC1SMN1; SMN2
SCHEMBL6206241 0.82 RAB9A (0.48) POLBRAB9AADORA2AALDH1A1MEN1
SCHEMBL6205208 0.82 CHRM3 (0.53) POLBRAB9AADORA2AALDH1A1MEN1
SCHEMBL6206374 0.80 ADORA2A (0.58) POLBRAB9AADORA2AALDH1A1MEN1
SCHEMBL6205245 0.79 HPGD (0.55) POLBRAB9AADORA2AALDH1A1NPC1
SCHEMBL6206694 0.79 WDR5 (0.47) POLBRAB9AADORA2A
SCHEMBL29050126 0.76 ALDH1A1 (0.60) POLBRAB9AALDH1A1MEN1KMT2A
SCHEMBL6205349 0.75 NHERF1 (0.65) POLBADORA2ASMN1; SMN2ADORA1
SCHEMBL6224870 0.75 CFTR (0.62) POLBRAB9AADORA2ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP claimed