SCHEMBL6207480

SCHEMBL6207480

CCc1c(C)c(C(=O)O)c[nH]c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
KDM3B Q7LBC6 2/20 0.41
DYRK1A Q13627 1/20 0.41
CSNK2A1 P68400 3/20 0.39
CSNK2A2 P19784 2/20 0.39
CSNK2B P67870 2/20 0.39
NOTUM Q6P988 2/20 0.38
GABRA1 P14867 2/20 0.38
GABRB2 P47870 2/20 0.38
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRA4 P48169 1/20 0.38
GABRE P78334 1/20 0.38
GABRA6 Q16445 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208722 0.86 KDM4E (0.44) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6207870 0.78 KDM4E (0.41) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6207236 0.77 DYRK1A (0.47) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6208699 0.77 KDM4E (0.43) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL27695803 0.76 HCAR2 (0.43) KDM4EKDM3BCSNK2A1CSNK2A2CSNK2B
SCHEMBL6206909 0.75 KDM4E (0.41) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6208037 0.74 DYRK1A (0.52) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL23674962 0.73 NAPRT (0.48) KDM4EKDM3BDYRK1AGABRA1GABRB2
SCHEMBL7121722 0.72 PRNP (0.38) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL10901788 0.71 GABRP (0.43) KDM4ECSNK2A1GABRA1GABRB2GABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546133-A2 N-SUBSTITUTE-2-OXODIHYDROPYRIDINE DERIVATIVES AS NPY ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2005-06-29 EP disclosed
WO-2004031175-A2 N-SUBSTITUTED-2-OXODIHYDROPYRIDINE DERIVATIVES AS NPY ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2004-04-15 WO disclosed