SCHEMBL6208699

SCHEMBL6208699

CCc1c(C(=O)O)c[nH]c(=O)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
KDM3B Q7LBC6 1/20 0.40
DYRK1A Q13627 1/20 0.40
HCAR2 Q8TDS4 1/20 0.38
CSNK2A1 P68400 3/20 0.36
CSNK2A2 P19784 2/20 0.36
CSNK2B P67870 2/20 0.36
NAPRT Q6XQN6 1/20 0.34
NOTUM Q6P988 1/20 0.33
HTT P42858 1/20 0.33
PIM3 Q86V86 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
HPGD P15428 2/20 0.33
GAA P10253 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PRKAB2 O43741 2/20 0.32
PRKAG1 P54619 2/20 0.32
PRKAA2 P54646 2/20 0.32
PRKAA1 Q13131 2/20 0.32
PRKAG3 Q9UGI9 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208722 0.81 KDM4E (0.44) KDM4EKDM3BDYRK1AHCAR2CSNK2A1
SCHEMBL6206909 0.80 KDM4E (0.41) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6207236 0.79 DYRK1A (0.47) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6207480 0.77 KDM4E (0.44) KDM4EKDM3BDYRK1AHCAR2CSNK2A1
SCHEMBL6207870 0.77 KDM4E (0.41) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL7121722 0.74 PRNP (0.38) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL26708623 0.73 DYRK1A (0.52) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL10760134 0.70 KDM4E (0.45) KDM4ECSNK2A1CSNK2A2CSNK2BHTT
SCHEMBL2655336 0.69 CES2 (0.45) KDM4EGAAMEN1ALDH1A1CYP1A2
SCHEMBL3718398 0.68 KDM4E (0.43) KDM4ECSNK2A1CSNK2A2CSNK2BHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546133-A2 N-SUBSTITUTE-2-OXODIHYDROPYRIDINE DERIVATIVES AS NPY ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2005-06-29 EP claimed
WO-2004031175-A2 N-SUBSTITUTED-2-OXODIHYDROPYRIDINE DERIVATIVES AS NPY ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2004-04-15 WO claimed
EP-1546133-A2 N-SUBSTITUTE-2-OXODIHYDROPYRIDINE DERIVATIVES AS NPY ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2005-06-29 EP disclosed
WO-2004031175-A2 N-SUBSTITUTED-2-OXODIHYDROPYRIDINE DERIVATIVES AS NPY ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2004-04-15 WO disclosed