SCHEMBL6208722

SCHEMBL6208722

CCc1c(C(=O)O)c[nH]c(=O)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
KDM3B Q7LBC6 1/20 0.41
DYRK1A Q13627 1/20 0.41
CSNK2A1 P68400 3/20 0.39
CSNK2A2 P19784 2/20 0.39
CSNK2B P67870 2/20 0.39
NOTUM Q6P988 2/20 0.38
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PIM3 Q86V86 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
NAPRT Q6XQN6 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
GABRA1 P14867 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6207480 0.86 KDM4E (0.44) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6208699 0.81 KDM4E (0.43) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6207236 0.81 DYRK1A (0.47) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6206909 0.78 KDM4E (0.41) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL7121722 0.76 PRNP (0.38) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL6207870 0.75 KDM4E (0.41) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL27695803 0.72 HCAR2 (0.43) KDM4EKDM3BCSNK2A1CSNK2A2CSNK2B
SCHEMBL10901788 0.71 GABRP (0.43) KDM4ECSNK2A1HPGDHSD17B10CYP1A2
SCHEMBL6208037 0.70 DYRK1A (0.52) KDM4EKDM3BDYRK1ACSNK2A1CSNK2A2
SCHEMBL27412755 0.69 KDM4E (0.42) KDM4ECSNK2A1NOTUMGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546133-A2 N-SUBSTITUTE-2-OXODIHYDROPYRIDINE DERIVATIVES AS NPY ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2005-06-29 EP disclosed
WO-2004031175-A2 N-SUBSTITUTED-2-OXODIHYDROPYRIDINE DERIVATIVES AS NPY ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 2004-04-15 WO disclosed