SCHEMBL6209310

SCHEMBL6209310

Brc1ccc([C]2CCCC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.44
ALDH1A1 P00352 7/20 0.43
MAPK1 P28482 2/20 0.43
HPGD P15428 2/20 0.41
HTR2C P28335 2/20 0.40
MAPT P10636 4/20 0.39
KMT2A Q03164 3/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
CASP3 P42574 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
GALR1 P47211 1/20 0.35
ALOX15 P16050 2/20 0.35
CA12 O43570 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208982 0.97 ALDH1A1 (0.44) CYP2A6ALDH1A1MAPK1HPGDHTR2C
SCHEMBL4326011 0.88 CYP2A6 (0.50) CYP2A6ALDH1A1MAPK1HPGDHTR2C
SCHEMBL21855095 0.78 CYP2A6 (0.44) CYP2A6ALDH1A1MAPK1HPGDHTR2C
SCHEMBL218474 0.72 LMNA (0.44) CYP2A6ALDH1A1HPGDHTR2CRAB9A
SCHEMBL2537130 0.72 MAPK14 (0.45) KMT2ARAB9ANPC1GALR1
SCHEMBL4555821 0.72 ALDH1A1 (0.53) ALDH1A1MAPK1HPGDMAPTKMT2A
SCHEMBL6100514 0.72 ACHE (0.44) ALDH1A1MAPK1HPGDMAPTGALR1
SCHEMBL8310754 0.72 TRPA1 (0.40) ALDH1A1
SCHEMBL1673427 0.71 ALDH1A1 (0.73) CYP2A6ALDH1A1MAPK1MAPTKMT2A
SCHEMBL68094 0.71 ALDH1A1 (0.73) CYP2A6ALDH1A1MAPK1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4118086-A1 COMPOUNDS USEFUL AS KINASE INHIBITORS Fochon Biosciences, Ltd. (CN) 2023-01-18 EP disclosed
WO-2021180107-A1 COMPOUNDS USEFUL AS KINASE INHIBITORS FOCHON PHARMACEUTICALS, LTD. (CN) 2021-09-16 WO disclosed
EP-1507763-A1 TETRAHYDROISOQUINOLINE DERIVATIVES Bayer HealthCare AG (DE) 2005-02-23 EP disclosed
WO-2003097607-A1 TETRAHYDROISOQUINOLINE DERIVATIVES BAYER HEALTHCARE AG (DE) 2003-11-27 WO disclosed