SCHEMBL8310754

SCHEMBL8310754

BrCc1ccc([C]2CCCCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
HRH3 Q9Y5N1 7/20 0.35
HRH4 Q9H3N8 2/20 0.35
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL679626 0.76 TSHR (0.56) TRPA1ALDH1A1TSHRHRH3HRH4
SCHEMBL9609757 0.76 TSHR (0.56) TRPA1ALDH1A1TSHRHRH3HRH4
SCHEMBL6208982 0.75 ALDH1A1 (0.44) ALDH1A1
Methane SCHEMBL11480910 0.73 TSHR (0.53) TRPA1ALDH1A1TSHRHRH3HRH4
Water SCHEMBL11481683 0.73 TSHR (0.53) TRPA1ALDH1A1TSHRHRH3HRH4
SCHEMBL9176921 0.73 NISCH (0.44) HRH3
SCHEMBL131361 0.72 ALDH1A1 (0.67) TRPA1ALDH1A1TSHRHRH3CES2
SCHEMBL6209310 0.72 CYP2A6 (0.44) ALDH1A1
SCHEMBL20272050 0.71 NISCH (0.41) ALDH1A1TSHR
SCHEMBL8885877 0.71 ACMSD (0.44) TRPA1ALDH1A1TSHRHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920424-A1 NON-PEPTIDE BOMBESIN RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1999-06-09 EP disclosed
WO-1998007718-A1 NON-PEPTIDE BOMBESIN RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1998-02-26 WO disclosed