SCHEMBL6209419

SCHEMBL6209419

O=C(NC(Cc1cccc(O)c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.42
CTSK P43235 3/20 0.42
HPGDS O60760 2/20 0.41
CTSL P07711 3/20 0.41
CTSB P07858 3/20 0.41
CTSS P25774 3/20 0.41
TAAR1 Q96RJ0 1/20 0.40
GPR132 Q9UNW8 4/20 0.39
PTAFR P25105 1/20 0.39
CTSV O60911 1/20 0.39
CMKLR2 P46091 1/20 0.38
CMKLR1 Q99788 1/20 0.38
ROCK2 O75116 1/20 0.36
SMYD3 Q9H7B4 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041541 0.92 CTSK (0.49) ACECTSKCTSLCTSSTAAR1
SCHEMBL4044160 0.91 CTSB (0.37) ACECTSKCTSBCTSSTAAR1
SCHEMBL6209046 0.86 CTSK (0.47) ACECTSKHPGDSCTSLCTSB
SCHEMBL4039023 0.85 CTSK (0.50) ACECTSKCTSSTAAR1GPR132
SCHEMBL4044930 0.84 DPP4 (0.38) SMYD3
SCHEMBL4047615 0.84 CTSB (0.38) ACECTSKCTSBCTSSTAAR1
SCHEMBL6213366 0.83 CTSK (0.42) CTSKHPGDSCTSLCTSBCTSS
SCHEMBL4041209 0.83 HPGDS (0.39) ACECTSKHPGDSCTSBCTSS
SCHEMBL4042537 0.83 CTSK (0.49) ACECTSKCTSLCTSBCTSS
SCHEMBL4041490 0.82 CTSK (0.51) ACECTSKCTSSSMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed