SCHEMBL4044160

SCHEMBL4044160

O=C(NC(Cc1cccc(O)c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
EPHX1 P07099 1/20 0.36
ACE P12821 2/20 0.35
FKBP1A P62942 1/20 0.35
GPR132 Q9UNW8 4/20 0.35
TAAR1 Q96RJ0 1/20 0.35
CHRNA7 P36544 1/20 0.35
CMKLR2 P46091 1/20 0.35
CMKLR1 Q99788 1/20 0.35
NAMPT P43490 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047615 0.93 CTSB (0.38) CTSBCTSSCTSKACEFKBP1A
SCHEMBL4047882 0.91 F2 (0.36) CTSBCTSSCTSKEPHX1ACE
SCHEMBL6209419 0.91 ACE (0.42) CTSBCTSSCTSKACEGPR132
SCHEMBL4045511 0.90 F2 (0.38) CTSBCTSSCTSK
SCHEMBL4050328 0.90 SCN9A (0.39) CTSBCTSSCTSKACEFKBP1A
SCHEMBL4045597 0.90 ACE (0.36) CTSBCTSSCTSKEPHX1ACE
SCHEMBL4046932 0.90 GPR132 (0.35) CTSBCTSSCTSKGPR132
SCHEMBL4043952 0.89 CTSK (0.42) CTSBCTSSCTSKFKBP1ACHRNA7
SCHEMBL4043998 0.88 FKBP1A (0.37) CTSBCTSSCTSKEPHX1FKBP1A
SCHEMBL4042165 0.87 EPHX1 (0.37) CTSBCTSSCTSKEPHX1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed