SCHEMBL6209727

SCHEMBL6209727

CC(CCNC(=O)c1ccc(Oc2ccccc2)cc1)CC(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 5/20 0.42
MMP13 P45452 2/20 0.41
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
CCR5 P51681 1/20 0.38
CTSK P43235 2/20 0.38
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.36
HTT P42858 1/20 0.36
MAPK14 Q16539 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RECQL P46063 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210327 0.93 GAA (0.45) CHRM4POLBHPGDCCR5GAA
SCHEMBL6210258 0.91 POLB (0.42) CHRM4MMP13POLBHPGDCCR5
SCHEMBL6210874 0.91 ALDH1A1 (0.40) CHRM4MMP13POLBHPGDCTSK
SCHEMBL6211027 0.90 NAMPT (0.40) CHRM4POLBHPGDCCR5CTSK
SCHEMBL6209043 0.90 LMNA (0.41) POLBCCR5CTSKLMNASMN1; SMN2
SCHEMBL6212088 0.89 SLC6A5 (0.40) CHRM4CCR5CTSKLMNAHTT
SCHEMBL6259636 0.88 HDAC3 (0.35) CHRM4POLBHPGDCTSKLMNA
SCHEMBL6213867 0.88 CHRM4 (0.40) CHRM4MMP13POLBHPGDCCR5
SCHEMBL6211167 0.87 CTSK (0.39) HPGDCTSKKMT2AHTTSMN1; SMN2
SCHEMBL6212722 0.87 CHRM4 (0.43) CHRM4MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed