SCHEMBL6209733

SCHEMBL6209733

COc1ccc(C(CN)CCc2ccccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.64
TSHR P16473 1/20 0.48
LTA4H P09960 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
POLB P06746 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
AOC3 Q16853 1/20 0.45
ABCB1 P08183 1/20 0.44
CNR2 P34972 1/20 0.44
MAPK1 P28482 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452354 0.84 ALDH1A1 (0.56) ALDH1A1TSHRLTA4HTAAR1POLB
SCHEMBL7412978 0.84 CASR (0.51) ALDH1A1TAAR1
SCHEMBL20052924 0.84 CASR (0.51) ALDH1A1TAAR1
SCHEMBL15286352 0.83 GABBR2 (0.50) TAAR1
SCHEMBL29048475 0.82 ALDH1A1 (0.43) ALDH1A1TAAR1L3MBTL1CNR2
SCHEMBL6211904 0.81 L3MBTL1 (0.55) ALDH1A1TSHRTAAR1L3MBTL1NPC1
SCHEMBL17996029 0.80 GABBR2 (0.47) TAAR1
SCHEMBL11079771 0.79 ALDH1A1 (0.54) ALDH1A1TSHRTAAR1L3MBTL1SLC6A2
SCHEMBL29048454 0.79 GABBR2 (0.51) TSHRTAAR1SLC6A2SLC6A4CNR2
SCHEMBL9872486 0.78 ALDH1A1 (0.51) ALDH1A1TSHRTAAR1L3MBTL1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050234096-A1 Tetrahydroisoquinoline derivatives BAYER HEALTHCARE AG (DE) 2005-10-20 US disclosed
US-6956040-B2 Oxazolidinone piperazinyl derivatives as potential antimicrobials RANBAXY LABORATORIES LIMITED (IN) 2005-10-18 US disclosed
EP-1507763-A1 TETRAHYDROISOQUINOLINE DERIVATIVES Bayer HealthCare AG (DE) 2005-02-23 EP disclosed
US-20040254162-A1 Oxazolidinone derivatives as antimicrobials RANBAXY LABORATORIES LIMITED (IN) 2004-12-16 US disclosed
WO-2003097607-A1 TETRAHYDROISOQUINOLINE DERIVATIVES BAYER HEALTHCARE AG (DE) 2003-11-27 WO disclosed
US-20030119817-A1 Oxazolidinone derivatives as potential antimicrobials MEHTA ANITA (IN) 2003-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030119817-A1 Oxazolidinone derivatives as potential antimicrobials OXA1L, PDK4, SDHA ALDH1A1 973/4885TSHR 1336/4885LTA4H 1714/4885
US-20040254162-A1 Oxazolidinone derivatives as antimicrobials PPARD, PDK4, OXA1L ALDH1A1 934/4885TSHR 1486/4885LTA4H 1947/4885
US-20050234096-A1 Tetrahydroisoquinoline derivatives PPARD, PPARG, PPARA ALDH1A1 2218/4885TSHR 1402/4885LTA4H 1239/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.