SCHEMBL6208880

SCHEMBL6208880

NC(=O)CCCC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 1/20 0.38
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.37
ITGB1 P05556 1/20 0.36
ITGAV P06756 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
FKBP1A P62942 1/20 0.36
GAA P10253 1/20 0.35
MAPK1 P28482 1/20 0.35
CHRM1 P11229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210370 0.86 FKBP1A (0.41) TSHRALDH1A1SMYD3CYP2C19FKBP1A
SCHEMBL6208973 0.86 TBXAS1 (0.35) HPGDALDH1A1MAPK1
SCHEMBL4038371 0.86 KDM4E (0.40) KDM4EHPGDTSHRHSD17B10ALDH1A1
SCHEMBL6208666 0.85 KDM4E (0.39) KDM4EHPGDTSHRHSD17B10ALDH1A1
SCHEMBL6208517 0.85 HSD17B10 (0.41) KDM4EHPGDTSHRHSD17B10ALDH1A1
SCHEMBL6209393 0.82 CTSL (0.36) SMYD3
SCHEMBL6211364 0.81 DPP4 (0.45) ALDH1A1SMYD3CYP3A4CYP2C19
SCHEMBL6212946 0.80 RAB9A (0.47) ALDH1A1SMYD3GAAMAPK1
SCHEMBL6212092 0.80 PREP (0.48) TSHRALDH1A1CYP3A4GAA
SCHEMBL5941964 0.80 PKM (0.38) TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed