SCHEMBL6218845

SCHEMBL6218845

COC(=O)C(CC(C)C)C(N1CCC(Oc2ccc(F)cc2Br)CC1)=S(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR6 P46095 12/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HRH1 P35367 1/20 0.36
CCR3 P51677 1/20 0.36
CYP2D6 P10635 1/20 0.36
IKBKB O14920 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6218909 0.91 IKBKB (0.38) GPR6HRH1CCR3IKBKB
SCHEMBL6218839 0.76 PTGDR (0.42) GPR6ALDH1A1L3MBTL1CYP2D6IKBKB
SCHEMBL6249262 0.76 IKBKB (0.42) GPR6ALDH1A1HTTL3MBTL1IKBKB
SCHEMBL6362089 0.75 PTGDR (0.41) GPR6ALDH1A1L3MBTL1CYP2D6IKBKB
SCHEMBL27623158 0.73 PKM (0.47) IKBKB
Hydrochloric Acid SCHEMBL2774596 0.72 DPP4 (0.48) GPR6IKBKB
SCHEMBL2773855 0.71 CCR1 (0.48) GPR6LMNAHRH1CCR3IKBKB
SCHEMBL6218902 0.71 PTGDR (0.42) GPR6ALDH1A1L3MBTL1IKBKB
SCHEMBL6104086 0.70 PTGDR (0.45) GPR6ALDH1A1HRH1CCR3IKBKB
SCHEMBL2773558 0.70 GPR119 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539159-A1 SULPHONYLPIPERIDINE DERIVATIVES CONTAINING AN ARYL OR HETEROARYL GROUP FOR USE AS MATRIX METALLOPROTEINASE INHIBITORS Astrazeneca AB (SE) 2005-06-15 EP disclosed
WO-2004006926-A1 SULPHONYLPIPERIDINE DERIVATIVES CONTAINING AN ARYL OR HETEROARYL GROUP FOR USE AS MATRIX METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2004-01-22 WO disclosed