SCHEMBL622356

SCHEMBL622356

COC(=O)CCCCC(=O)N[C@H](C(=O)NC(C=O)Cc1ccc(O)cc1)C(C)C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSB P07858 2/20 0.45
GRIA1 P42261 7/20 0.41
REN P00797 1/20 0.40
CTSD P07339 1/20 0.40
CNR1 P21554 1/20 0.39
CHRNA1 P02708 1/20 0.38
CHRNG P07510 1/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
GRIN1 Q05586 1/20 0.38
CHRND Q07001 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRM1 Q13255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL621504 0.99 CTSB (0.44) CTSBGRIA1CNR1
SCHEMBL10084885 0.91 CASP1 (0.46) CTSBCTSD
SCHEMBL622823 0.90 CTSB (0.54) CTSBCTSD
SCHEMBL622452 0.90 CASP1 (0.45) CTSBCTSDCNR1
SCHEMBL622810 0.89 CTSB (0.53) CTSBCTSD
SCHEMBL623329 0.88 CTSB (0.54) CTSBCTSD
SCHEMBL10084886 0.87 ITGB3 (0.48)
SCHEMBL622149 0.86 CTSB (0.51) CTSB
SCHEMBL10085515 0.86 ITGB3 (0.50)
SCHEMBL623355 0.86 ITGB3 (0.39) CTSBCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed