SCHEMBL622452

SCHEMBL622452

COC(=O)CCCCCCC(=O)N[C@H](C(=O)NC(C=O)Cc1ccc(OC)cc1)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.45
ALDH1A1 P00352 2/20 0.43
KMT2A Q03164 1/20 0.42
CTSB P07858 2/20 0.41
CNR1 P21554 2/20 0.39
CTSD P07339 3/20 0.39
CTSK P43235 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.38
HDAC2 Q92769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10084885 0.99 CASP1 (0.46) CASP1ALDH1A1KMT2ACTSBCTSD
SCHEMBL621504 0.91 CTSB (0.44) CTSBCNR1
SCHEMBL10085515 0.90 ITGB3 (0.50)
SCHEMBL623355 0.90 ITGB3 (0.39) CASP1CTSBCTSD
SCHEMBL622810 0.90 CTSB (0.53) CTSBCTSDCTSK
SCHEMBL622356 0.90 CTSB (0.45) CTSBCNR1CTSD
SCHEMBL10084886 0.89 ITGB3 (0.48)
SCHEMBL622823 0.89 CTSB (0.54) CTSBCTSDCTSK
SCHEMBL623001 0.88 CTSB (0.50) CTSB
SCHEMBL622149 0.87 CTSB (0.51) CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed