SCHEMBL622532

SCHEMBL622532

COC(=O)CCCCC(=O)N[C@H](C(=O)NC(Cc1ccccc1)C(=O)C(=O)NC1CC1)C(C)C

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 7/20 0.55
EPHX2 P34913 2/20 0.44
HRH1 P35367 3/20 0.42
CASP1 P29466 1/20 0.42
CTSD P07339 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623798 0.99 CAPN1 (0.54) CAPN1EPHX2HRH1
SCHEMBL621465 0.84 CAPN1 (0.52) CAPN1CASP1CTSD
SCHEMBL621544 0.83 CTSD (0.45) EPHX2CTSD
SCHEMBL621481 0.82 CAPN1 (0.67) CAPN1HRH1
SCHEMBL621480 0.82 CAPN1 (0.67) CAPN1HRH1
SCHEMBL623310 0.81 CASP1 (0.47) CASP1CTSD
SCHEMBL622809 0.80 HDAC1 (0.48) CASP1CTSD
SCHEMBL23921539 0.78 GPR139 (0.56) CAPN1CTSD
SCHEMBL21526187 0.78 GPR139 (0.56) CAPN1CTSD
SCHEMBL21555036 0.78 GPR139 (0.56) CAPN1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed