SCHEMBL6228641

SCHEMBL6228641

Cc1cc(CCNc2ccccc2)ccc1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.53
ERCC1 P07992 2/20 0.52
ERCC4 Q92889 2/20 0.52
ESR1 P03372 2/20 0.50
ESR2 Q92731 2/20 0.50
STAT6 P42226 1/20 0.46
GFER P55789 2/20 0.46
POLB P06746 1/20 0.46
KMT2A Q03164 1/20 0.46
MAPT P10636 5/20 0.45
MAPK1 P28482 2/20 0.45
ALOX15 P16050 2/20 0.45
HIF1A Q16665 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.45
TSHR P16473 1/20 0.45
NFKB1 P19838 1/20 0.45
THPO P40225 1/20 0.45
ADRB2 P07550 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410353 0.85 ERCC1 (0.68) L3MBTL1ERCC1ERCC4GFERPOLB
SCHEMBL19842170 0.80 CNR1 (0.61) ERCC1ERCC4KMT2AMAPTTP53
Hydrochloric Acid SCHEMBL5310916 0.79 L3MBTL1 (0.56) L3MBTL1ERCC1ERCC4GFERPOLB
SCHEMBL172708 0.79 ESR1 (0.61) ESR1ESR2ALOX15TP53ADRB2
SCHEMBL12305680 0.78 MAPT (0.72) ESR1ESR2GFERPOLBMAPT
SCHEMBL11276210 0.77 L3MBTL1 (0.53) L3MBTL1ERCC1ERCC4GFERPOLB
SCHEMBL6184638 0.77 MAPT (0.58) ERCC1ERCC4ESR1ESR2GFER
SCHEMBL10055000 0.76 L3MBTL1 (0.86) L3MBTL1MAPTCYP1A2TSHRNFKB1
SCHEMBL1924746 0.76 ESR1 (0.74) ESR1ESR2MAPTMAPK1ALOX15
SCHEMBL29720481 0.76 ESR1 (0.74) ESR1ESR2MAPTMAPK1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562595-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2005-08-17 EP disclosed
WO-2004026305-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST ELI LILLY AND COMPANY (US) 2004-04-01 WO disclosed