SCHEMBL623002

SCHEMBL623002

COC(=O)CCCCCCC(=O)N[C@H](C(=O)NC(C=O)Cc1ccc(OCC(=O)OC(C)(C)C)cc1)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTRA1 Q92743 3/20 0.40
HDAC8 Q9BY41 3/20 0.39
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
REN P00797 4/20 0.36
CTSB P07858 1/20 0.36
KLK5 Q9Y337 1/20 0.36
CTSD P07339 2/20 0.35
ACACB O00763 1/20 0.35
PTPN1 P18031 1/20 0.35
CASP1 P29466 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623355 0.87 ITGB3 (0.39) HDAC8ITGB3ITGA2BCTSBCTSD
SCHEMBL10085515 0.87 ITGB3 (0.50) ITGB3ITGA2BACACB
SCHEMBL622452 0.86 CASP1 (0.45) CTSBCTSDCASP1
SCHEMBL10084886 0.86 ITGB3 (0.48) ITGB3ITGA2BACACB
SCHEMBL10084885 0.85 CASP1 (0.46) CTSBCTSDCASP1
SCHEMBL623001 0.84 CTSB (0.50) CTSB
SCHEMBL621504 0.83 CTSB (0.44) CTSB
SCHEMBL622149 0.83 CTSB (0.51) CTSB
SCHEMBL622810 0.82 CTSB (0.53) CTSBCTSD
SCHEMBL622356 0.82 CTSB (0.45) RENCTSBCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed