SCHEMBL6233812

SCHEMBL6233812

Cc1ccc(S(=O)(=O)OCCCCC#Cc2cncc(OC(C(=O)OC(C)(C)C)[C@@H]3CCCN3)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 12/20 0.37
CHRNA3 P32297 8/20 0.37
CHRNA4 P43681 5/20 0.37
CHRNA2 Q15822 5/20 0.37
CHRNB4 P30926 4/20 0.37
CHRNB1 P11230 1/20 0.30
CHRNB3 Q05901 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6231761 0.96 CHRNB2 (0.40) CHRNB2CHRNA3CHRNA4CHRNA2CHRNB4
SCHEMBL5802609 0.85 FKBP1A (0.36) CHRNB2
SCHEMBL6233687 0.81 CHRNB2 (0.56) CHRNB2CHRNA3CHRNA4CHRNA2CHRNB4
SCHEMBL8149383 0.80 CHRNB2 (0.46) CHRNB2CHRNA3CHRNA4CHRNA2CHRNB4
SCHEMBL6273656 0.80 CHRNB2 (0.46) CHRNB2CHRNA3CHRNA4CHRNA2CHRNB4
SCHEMBL8506415 0.80 CHRNB2 (0.46) CHRNB2CHRNA3CHRNA4CHRNA2CHRNB4
SCHEMBL2498122 0.75 CHRNA3 (0.51) CHRNB2CHRNA3CHRNA4CHRNA2CHRNB4
SCHEMBL2500469 0.75 CHRNB2 (0.46) CHRNB2CHRNA3CHRNA4CHRNA2CHRNB4
SCHEMBL8911083 0.72 MMP13 (0.38)
SCHEMBL5806257 0.71 NPC1 (0.35) CHRNB2CHRNA3CHRNA4CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005000806-A2 LIGANDS FOR NICOTINIC ACETYLCHOLINE RECEPTORS, AND METHODS OF MAKING AND USING THEM GEORGETOWN UNIVERSITY (US) 2005-01-06 WO disclosed