SCHEMBL6234787

SCHEMBL6234787

COc1ccccc1COCCNCCN

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 14/20 0.57
HTR1A P08908 1/20 0.55
ADRA1D P25100 1/20 0.55
ADRA1A P35348 1/20 0.55
ADRA1B P35368 1/20 0.55
BCHE P06276 5/20 0.53
ACHE P22303 5/20 0.53
CHRM4 P08173 5/20 0.53
CHRM5 P08912 5/20 0.53
CHRM1 P11229 5/20 0.53
CHRM3 P20309 5/20 0.53
GRIN1 Q05586 4/20 0.53
GRIN2A Q12879 4/20 0.53
RECQL P46063 2/20 0.53
TP53 P04637 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
TSHR P16473 1/20 0.53
THPO P40225 1/20 0.53
IDO1 P14902 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237597 0.81 CHRM2 (0.47) CHRM2HTR1AADRA1DADRA1AADRA1B
SCHEMBL6234780 0.80 HTR1A (0.47) CHRM2HTR1AADRA1DADRA1AADRA1B
SCHEMBL4918374 0.80 CHRM2 (0.80) CHRM2BCHEACHECHRM4CHRM5
SCHEMBL4918894 0.80 CHRM2 (0.80) CHRM2BCHEACHECHRM4CHRM5
SCHEMBL4918881 0.80 CHRM2 (0.80) CHRM2BCHEACHECHRM4CHRM5
SCHEMBL4909317 0.79 CHRM2 (0.79) CHRM2BCHEACHECHRM4CHRM5
SCHEMBL6244580 0.78 IDO1 (0.49) CHRM2HTR1AADRA1DADRA1AADRA1B
SCHEMBL10458199 0.77 IDO1 (0.56) CHRM2HTR1AADRA1DADRA1AADRA1B
SCHEMBL28384840 0.77 IDO1 (0.66) CHRM2CHRM1GRIN1GRIN2AIDO1
SCHEMBL26654 0.76 IDO1 (0.69) CHRM2BCHEACHECHRM1GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005011697-A2 SULFONAMIDE DERIVATIVES WITH ACTIVITY ON PROTEIN KINASE A AND B ASTEX THERAPEUTICS LIMITED (GB) 2005-02-10 WO disclosed