SCHEMBL6234853

SCHEMBL6234853

Cc1ccc2sc(N)nc2c1C

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
HSD17B10 Q99714 1/20 0.52
CYP3A4 P08684 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 3/20 0.47
PDPK1 O15530 1/20 0.47
PDE10A Q9Y233 1/20 0.47
TP53 P04637 2/20 0.46
TSHR P16473 1/20 0.46
RAB9A P51151 2/20 0.45
NPC1 O15118 1/20 0.45
GAA P10253 1/20 0.44
HTT P42858 1/20 0.43
MAPT P10636 4/20 0.43
NSD1 Q96L73 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754543 1.00 ALDH1A1 (0.61) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2
SCHEMBL30829728 0.81 SMN1; SMN2 (0.62) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2
SCHEMBL11718702 0.81 LMNA (0.58) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2
SCHEMBL30829749 0.81 LMNA (0.58) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2
SCHEMBL24425191 0.81 SMN1; SMN2 (0.62) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2
SCHEMBL23043060 0.81 ALDH1A1 (0.58) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2
SCHEMBL7936559 0.81 PDPK1 (0.58) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2
SCHEMBL6118333 0.80 SMN1; SMN2 (0.59) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2
SCHEMBL12109863 0.79 NPC1 (0.49) ALDH1A1HSD17B10TDP1SMN1; SMN2LMNA
SCHEMBL25081101 0.78 ALDH1A1 (0.54) ALDH1A1HSD17B10CYP3A4TDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3759111-A1 PHARMACEUTICAL COMPOUNDS Otsuka Pharmaceutical Co., Ltd. (JP) 2021-01-06 EP claimed
EP-1178977-B1 ION CHANNEL MODULATING AGENTS NEUROSEARCH AS (DK) 2005-06-01 EP claimed
US-6759422-B2 ADMINISTERING BENZOTHIAZOLE COMPOUND FOR THERAPY, PROPHYLAXIS OF DISEASE NEUROSEARCH A/S (DK) 2004-07-06 US claimed
WO-2004039409-A2 COMPOSITION COMPRISING ACTIVATORS OF IK POTASSIUM CHANNELS AND CALCINEURIN ANTAGONISTS AND USE THEREOF SWITCH BIOTECH AG (DE) 2004-05-13 WO claimed
US-20030008906-A1 Ion channel modulating agents NEUROSEARCH A/S 2003-01-09 US claimed
US-20020061914-A1 Ion channel modulating agents NEUROSEARCH A/S (DK) 2002-05-23 US claimed
EP-1178977-A1 ION CHANNEL MODULATING AGENTS NEUROSEARCH A/S (DK) 2002-02-13 EP claimed
WO-2000069838-A1 ION CHANNEL MODULATING AGENTS NEUROSEARCH A/S (DK) 2000-11-23 WO claimed
US-20250382273-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INST NAT SANTE RECH MED (FR) 2025-12-18 US disclosed
EP-4460500-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2024-11-13 EP disclosed
CN-118660885-A Norbornene analogs and their use as potentiators of antitubercular drugs 国家医疗保健研究所 2024-09-17 CN disclosed
WO-2023131649-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-07-13 WO disclosed
EP-3294728-A1 SUBSTITUTED QUINOXALINE DERIVATIVES SELVITA S.A. (PL) 2018-03-21 EP disclosed
WO-2016180537-A1 SUBSTITUTED QUINOXALINE DERIVATIVES SELVITA S.A. (PL) 2016-11-17 WO disclosed
WO-2000069838-A1 ION CHANNEL MODULATING AGENTS NEUROSEARCH A/S (DK) 2000-11-23 WO disclosed
US-4086241-A Benzothiazolylimidazolidinone esters of furyl and thienyl substituted acids VELSICOL CHEMICAL CORPORATION (US) 1978-04-25 US disclosed
US-4055569-A HERBICIDE VELSICOL CHEMICAL CORPORATION (US) 1977-10-25 US disclosed
US-4054574-A HERBICIDES VELSICOL CHEMICAL CORPORATION (US) 1977-10-18 US disclosed
US-4045446-A 1-Benzothiazolyl-5-pyridylcarbonyloxyimidazolidinones VELSICOL CHEMICAL CORPORATION (US) 1977-08-30 US disclosed
US-4029491-A HERBICIDES VELSICOL CHEMICAL CORPORATION (US) 1977-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250382273-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS BBOX1, NDUFB6, NDUFB5 ALDH1A1 108/4885HSD17B10 227/4885CYP3A4 343/4885
US-20020061914-A1 Ion channel modulating agents KCNN1, KCNJ2, KCNN2 ALDH1A1 4274/4885HSD17B10 3867/4885CYP3A4 3663/4885
US-20030008906-A1 Ion channel modulating agents KCNN1, KCNJ2, KCNN2 ALDH1A1 4208/4885HSD17B10 3762/4885CYP3A4 3654/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.