SCHEMBL6237142

SCHEMBL6237142

COc1ccccc1N1CCN(CCCC(=O)CCCC(=O)O)CC1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.65
POLB P06746 1/20 0.65
HTR1A P08908 4/20 0.65
DRD2 P14416 5/20 0.65
HTR2A P28223 1/20 0.65
KDM4E B2RXH2 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
DRD3 P35462 2/20 0.63
ADRA1D P25100 3/20 0.63
ADRA1A P35348 1/20 0.63
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
HTR7 P34969 1/20 0.62
DRD4 P21917 1/20 0.62
ADRA1B P35368 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1491175 0.95 HTR1A (0.71) ALDH1A1POLBHTR1ADRD2HTR2A
SCHEMBL11030623 0.90 HTR1A (0.73) ALDH1A1HTR1ADRD2HTR2AKDM4E
SCHEMBL3160665 0.87 HTR1A (0.79) ALDH1A1HTR1ADRD2HTR2AKDM4E
Benzene SCHEMBL10433203 0.87 HTR1A (0.79) ALDH1A1HTR1ADRD2HTR2AKDM4E
SCHEMBL6238933 0.85 DRD2 (0.72) HTR1ADRD2DRD3ADRA1AHTR7
SCHEMBL21673062 0.85 ADRA1D (0.65) ALDH1A1HTR1ADRD2HTR2AKDM4E
SCHEMBL3188003 0.85 ALDH1A1 (0.71) ALDH1A1POLBHTR1ADRD2HTR2A
SCHEMBL15743486 0.84 HTR1A (0.67) ALDH1A1POLBHTR1ADRD2HTR2A
Hydrochloric Acid SCHEMBL3196115 0.84 HTR1A (0.71) ALDH1A1POLBHTR1ADRD2HTR2A
Valeric Acid SCHEMBL11081888 0.82 DRD2 (0.64) ALDH1A1HTR1ADRD2HTR2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005018643-A1 METABOLITES OF 1-{3-4`4-(2-METHOXYPHENYL) PIPERAZIN-1-YL!-PROPYL}-PIPERIDINE-2, 6-DIONE FOR USE IN THE TREATMENT OF BENIGN PROSTATIC HYPERPLASIA RANBAXY LABORATORIES LIMITED (IN) 2005-03-03 WO disclosed