SCHEMBL6237643

SCHEMBL6237643

N#CN1CCN(c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.51
CA9 Q16790 2/20 0.51
CA12 O43570 1/20 0.51
AKR1C3 P42330 1/20 0.49
DHFR P00374 1/20 0.46
ME2 P23368 1/20 0.43
ME1 P48163 1/20 0.43
ME3 Q16798 1/20 0.43
KDM4E B2RXH2 1/20 0.43
TP53 P04637 1/20 0.43
MLYCD O95822 1/20 0.43
NOTUM Q6P988 1/20 0.42
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42
DRD3 P35462 1/20 0.42
CYP3A4 P08684 2/20 0.41
NAAA Q02083 1/20 0.41
PHGDH O43175 2/20 0.40
CA1 P00915 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28650484 0.84 CA12 (0.65) CA2CA9CA12AKR1C3DHFR
SCHEMBL5535690 0.82 CA12 (0.55) CA2CA9CA12AKR1C3DHFR
SCHEMBL3712914 0.80 ALDH1A1 (0.60) TP53CYP3A4
SCHEMBL17513744 0.78 DRD2 (0.48) CA2CA9CA12AKR1C3ME2
SCHEMBL28842325 0.77 CA12 (0.56) CA2CA9CA12AKR1C3DHFR
SCHEMBL13285321 0.77 CA12 (0.56) CA2CA9CA12AKR1C3DHFR
SCHEMBL25075457 0.76 CA12 (0.45) CA2CA9CA12AKR1C3DHFR
SCHEMBL21542324 0.76 NOTUM (0.50) CA2CA9CA12AKR1C3DHFR
SCHEMBL6235020 0.76 NOTUM (0.48) KDM4ETP53NOTUMCYP3A4
SCHEMBL5536334 0.76 ME2 (0.66) CA2CA9CA12AKR1C3DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO claimed
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed