SCHEMBL6231959

SCHEMBL6231959

FC(F)(F)c1cc(Cl)cc(Nc2ncco2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 3/20 0.49
HDAC3 O15379 2/20 0.47
HDAC1 Q13547 2/20 0.47
HDAC2 Q92769 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
SLC13A3 Q8WWT9 1/20 0.38
NOTUM Q6P988 1/20 0.37
SCN9A Q15858 2/20 0.36
ALOX5 P09917 1/20 0.36
BRAF P15056 1/20 0.36
RAPGEF3 O95398 3/20 0.35
JUN P05412 3/20 0.35
NFKB1 P19838 3/20 0.35
NFKB2 Q00653 3/20 0.35
RELA Q04206 3/20 0.35
GRM4 Q14833 1/20 0.35
AURKA O14965 1/20 0.34
PIK3CG P48736 1/20 0.34
XPO1 O14980 1/20 0.34
ATF1 P18846 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237657 0.77 AURKA (0.57) RAPGEF4NFKB1GRM4AURKA
SCHEMBL30041659 0.76 EPHX2 (0.48) SCN9A
SCHEMBL6237353 0.74 RAPGEF4 (0.49) RAPGEF4GRM4
SCHEMBL17403481 0.72 RAPGEF4 (0.46) RAPGEF4HDAC3HDAC1HDAC2HDAC6
SCHEMBL6240725 0.72 TDO2 (0.51) BRAFGRM4
SCHEMBL6236093 0.70 CDK4 (0.40) SCN9ABRAF
SCHEMBL16014245 0.68 HDAC3 (0.48) RAPGEF4HDAC3HDAC1HDAC2HDAC6
SCHEMBL4374429 0.68 RAPGEF4 (0.53) RAPGEF4HDAC3HDAC1HDAC2HDAC6
SCHEMBL12706897 0.68 RAPGEF4 (0.57) RAPGEF4HDAC3HDAC1HDAC2HDAC6
Hydrochloric Acid SCHEMBL4376336 0.66 RAPGEF4 (0.51) RAPGEF4HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed