SCHEMBL6238748

SCHEMBL6238748

[CH]NC(=O)c1ccncc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.67
KDM4E B2RXH2 2/20 0.61
MPO P05164 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
ADORA3 P0DMS8 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2A6 P11509 1/20 0.61
CYP2C19 P33261 1/20 0.61
GAA P10253 1/20 0.59
TP53 P04637 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.54
HTT P42858 1/20 0.53
NAPRT Q6XQN6 1/20 0.52
CA1 P00915 1/20 0.52
CA9 Q16790 1/20 0.52
TSHR P16473 1/20 0.52
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
PTGS2 P35354 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004792 0.80 ALDH1A1 (0.73) ALDH1A1KDM4EMPOCYP1A2CYP3A4
SCHEMBL2992964 0.80 ALDH1A1 (1.00) ALDH1A1KDM4EMPOCYP1A2CYP3A4
SCHEMBL2998145 0.78 HDAC6 (0.76) ALDH1A1KDM4EMPOCYP1A2CYP3A4
Isoniazid SCHEMBL28211874 0.77 KDM4E (0.91) ALDH1A1KDM4EMPOCYP1A2CYP3A4
SCHEMBL8150076 0.76 ALDH1A1 (0.67) ALDH1A1KDM4EMPOCYP1A2CYP3A4
SCHEMBL1744086 0.76 ALDH1A1 (0.67) ALDH1A1KDM4EMPOCYP1A2CYP3A4
Isoniazid SCHEMBL228 0.76 KDM4E (1.00) ALDH1A1KDM4EMPOCYP1A2CYP3A4
Isoniazid SCHEMBL12264081 0.76 KDM4E (1.00) ALDH1A1KDM4EMPOCYP1A2CYP3A4
Isoniazid SCHEMBL16642160 0.76 KDM4E (1.00) ALDH1A1KDM4EMPOCYP1A2CYP3A4
Isoniazid SCHEMBL2390873 0.76 KDM4E (1.00) ALDH1A1KDM4EMPOCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019177-A1 AMINOPIPERIDINE AMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO claimed
WO-2005019177-A1 AMINOPIPERIDINE AMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed