SCHEMBL6239020

SCHEMBL6239020

NC(=O)c1ccc(-c2ccccc2)c(S(N)(=O)=O)c1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.49
IKBKB O14920 8/20 0.46
CHUK O15111 6/20 0.46
CA12 O43570 6/20 0.41
CA1 P00915 6/20 0.41
CA2 P00918 6/20 0.41
CA7 P43166 4/20 0.41
CA13 Q8N1Q1 4/20 0.41
CA9 Q16790 2/20 0.39
KAT6A Q92794 1/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
IKBKE Q14164 1/20 0.37
PKMYT1 Q99640 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534063 0.89 CA1 (0.42) BCAT2IKBKBCHUKCA12CA1
SCHEMBL8533060 0.85 SLC9A1 (0.40) BCAT2IKBKBCHUKCA12CA1
SCHEMBL23573105 0.80 BCAT2 (0.58) BCAT2IKBKBCHUKKAT6AKDM4E
SCHEMBL30903647 0.80 BCAT2 (0.62) BCAT2IKBKBCHUKCA12CA1
SCHEMBL17593027 0.80 BCAT2 (0.62) BCAT2IKBKBCHUKCA12CA1
SCHEMBL4101964 0.78 CA1 (0.33) BCAT2CA12CA1CA2CA7
SCHEMBL6239022 0.78 CA12 (0.46) CA12CA1CA2CA7CA13
SCHEMBL18816701 0.76 BCAT2 (0.53) BCAT2IKBKBCHUKPTGS1PTGS2
SCHEMBL8529538 0.74 PTGS2 (0.41) KAT6APTGS1PTGS2MAPTHPGD
SCHEMBL15925025 0.74 CA12 (0.42) CA12CA1CA2CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539686-A1 INHIBITORS OF FACTOR XA AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION CASCADE WARNER-LAMBERT COMPANY LLC (US) 2005-06-15 EP claimed
WO-2004024679-A1 INHIBITORS OF FACTOR XA AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION CASCADE WARNER-LAMBERT COMPANY LLC (US) 2004-03-25 WO claimed
EP-1539686-A1 INHIBITORS OF FACTOR XA AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION CASCADE WARNER-LAMBERT COMPANY LLC (US) 2005-06-15 EP disclosed
WO-2004024679-A1 INHIBITORS OF FACTOR XA AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION CASCADE WARNER-LAMBERT COMPANY LLC (US) 2004-03-25 WO disclosed