SCHEMBL623944

SCHEMBL623944

c1cn2nc(N3CCOCC3)sc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.40
RAB9A P51151 7/20 0.40
NPC1 O15118 5/20 0.40
AR P10275 3/20 0.38
ALOX15 P16050 2/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
MAPT P10636 5/20 0.37
TP53 P04637 3/20 0.37
USP2 O75604 1/20 0.37
PKM P14618 1/20 0.37
POLB P06746 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
THRB P10828 1/20 0.37
LMNA P02545 1/20 0.36
GAA P10253 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624035 0.73 SMN1; SMN2 (0.40) SMN1; SMN2RAB9ANPC1ARALOX15
SCHEMBL624034 0.70 LMNA (0.48) MAPTTP53POLBRXFP1THRB
SCHEMBL29930378 0.69 GPX4 (0.33)
SCHEMBL11005420 0.67 PIK3CA (0.45) PIK3CDPIK3CAPIK3CBMAPTTP53
SCHEMBL2305450 0.67 SMN1; SMN2 (0.48) SMN1; SMN2RAB9ANPC1ARALOX15
SCHEMBL625650 0.67 PIK3CA (0.39) SMN1; SMN2RAB9ANPC1ARPIK3CA
SCHEMBL1932306 0.66 NPC1 (0.53) SMN1; SMN2RAB9ANPC1ARPIK3CA
SCHEMBL11005416 0.65 RXFP1 (0.61) MAPTTP53POLBRXFP1THRB
SCHEMBL2750222 0.65 SMN1; SMN2 (0.49) SMN1; SMN2RAB9ANPC1ARALOX15
SCHEMBL2585764 0.63 SMPD3 (0.47) SMN1; SMN2RAB9ANPC1PIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed