SCHEMBL6239508

SCHEMBL6239508

CC(Br)C(=O)N(C)C1=C(Cl)C(=O)c2ccccc2C1=O.CN(C(=O)CBr)C1=C(Cl)C(=O)c2ccccc2C1=O.O=C(CBr)NC1=C(Cl)C(=O)c2ccccc2C1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.48
PAX8 Q06710 1/20 0.48
HKDC1 Q2TB90 1/20 0.48
TLR9 Q9NR96 1/20 0.48
HSP90AA1 P07900 2/20 0.44
HSP90AB1 P08238 2/20 0.44
MAPT P10636 8/20 0.38
ALDH1A1 P00352 6/20 0.38
HTT P42858 6/20 0.38
RAB9A P51151 4/20 0.38
NPSR1 Q6W5P4 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
ATM Q13315 2/20 0.38
LMNA P02545 4/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HPGD P15428 2/20 0.38
KDM4E B2RXH2 2/20 0.38
CDC25A P30304 3/20 0.38
TDP1 Q9NUW8 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6240574 0.93 TDP2 (0.55) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL6244227 0.81 MAOA (0.48) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL6241764 0.81 MAOA (0.51) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL6239428 0.79 HKDC1 (0.68) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL6240578 0.76 HSP90AA1 (0.52) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL6239513 0.75 HSP90AA1 (0.50) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL6240168 0.71 HKDC1 (0.43) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL6192892 0.70 MAOA (0.52) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL7957003 0.69 HKDC1 (0.78) TDP2PAX8HKDC1TLR9HSP90AA1
SCHEMBL10891344 0.67 HKDC1 (0.70) TDP2PAX8HKDC1TLR9HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016264-A2 DIAMINE DERIVATIVES OF QUINONE AND USES THEREOF AVALON PHARMACEUTICALS (US) 2005-02-24 WO disclosed