SCHEMBL6239608

SCHEMBL6239608

COc1ccccc1Nc1nc(C#N)nc(N2CCN(C(=O)OC(C)(C)C)CC2)n1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.47
GBA1 P04062 5/20 0.47
ALK Q9UM73 5/20 0.46
CTSL P07711 3/20 0.45
CTSB P07858 3/20 0.45
CTSS P25774 3/20 0.45
CTSK P43235 3/20 0.45
ACHE P22303 1/20 0.43
EGFR P00533 2/20 0.43
TLR9 Q9NR96 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
SLC2A1 P11166 1/20 0.42
PTPN11 Q06124 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236029 0.87 GPR119 (0.44) NSD2ALKCTSLCTSBCTSS
SCHEMBL6234182 0.86 MAPT (0.53) GBA1ALKACHEEGFR
SCHEMBL6239744 0.82 GBA1 (0.63) GBA1CTSLCTSBCTSSCTSK
SCHEMBL6238044 0.81 GBA1 (0.62) GBA1CTSLCTSBCTSSCTSK
SCHEMBL6239397 0.81 GBA1 (0.62) GBA1CTSLCTSBCTSSCTSK
SCHEMBL6238470 0.80 CTSS (0.68) GBA1CTSLCTSBCTSSCTSK
SCHEMBL6237209 0.80 CTSK (0.67) GBA1CTSLCTSBCTSSCTSK
SCHEMBL6238645 0.79 GBA1 (0.51) GBA1CTSLCTSBCTSSCTSK
SCHEMBL6272121 0.77 GBA1 (0.50) NSD2GBA1ALKCTSLCTSB
SCHEMBL6242579 0.77 GBA1 (0.50) GBA1CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005011703-A1 2-CYANO-1,3,5-TRIAZINE-4,6-DIAMINE DERIVATIVES AKZO NOBEL N.V. (NL) 2005-02-10 WO disclosed