SCHEMBL6243783

SCHEMBL6243783

Cc1cc2c(c(O)c1-c1ccc(C(=O)c3ccccc3C(=O)O)cc1)C(C)(C)CCC2(C)C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HNF4A P41235 3/20 0.60
RXRA P19793 11/20 0.53
RARG P13631 6/20 0.53
RARB P10826 5/20 0.53
RARA P10276 4/20 0.53
RXRB P28702 2/20 0.53
RXRG P48443 2/20 0.53
CDC25B P30305 1/20 0.46
ATM Q13315 1/20 0.46
ALDH1A1 P00352 1/20 0.45
AKR1C3 P42330 1/20 0.45
KMT2A Q03164 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
MEN1 O00255 1/20 0.43
CYP26A1 O43174 1/20 0.43
ABCB11 O95342 1/20 0.43
ESR1 P03372 1/20 0.43
PGR P06401 1/20 0.43
HTR1A P08908 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6244136 0.81 RXRA (0.62) RXRARARGRARBRARARXRB
SCHEMBL6242159 0.78 HNF4A (0.48) HNF4ARXRARARGRARBRARA
SCHEMBL6236530 0.77 RXRA (0.57) HNF4ARXRARARGRARBRARA
SCHEMBL6236924 0.77 CDC25B (0.59) HNF4ARXRARARGRARBRARA
SCHEMBL6901726 0.76 RXRA (0.69) RXRARARGRARBRARARXRB
SCHEMBL6242642 0.74 HNF4A (0.68) HNF4ARXRARARGRARBRARA
SCHEMBL9551769 0.74 HNF4A (0.55) HNF4ARXRARARGRARBRARA
SCHEMBL2128581 0.73 RXRA (0.68) RXRARARGRARBRARARXRB
SCHEMBL29440075 0.73 RXRA (0.68) RXRARARGRARBRARARXRB
SCHEMBL292500 0.73 RXRA (0.83) HNF4ARXRARARGRARBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005017185-A2 HEPATOCYTE NUCLEAR FACTOR 4α MODULATOR COMPOUNDS LIGAND PHARMCEUTICALS INCORPORATED (US) 2005-02-24 WO claimed
WO-2005017185-A2 HEPATOCYTE NUCLEAR FACTOR 4α MODULATOR COMPOUNDS LIGAND PHARMCEUTICALS INCORPORATED (US) 2005-02-24 WO disclosed