SCHEMBL623998

SCHEMBL623998

CCOC(=O)C1CCCN(c2nn3c(-c4cccc(OC(F)(F)F)c4)cnc3s2)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 13/20 0.51
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 2/20 0.45
HSD17B10 Q99714 2/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
FLT3 P36888 2/20 0.44
KCNH2 Q12809 2/20 0.44
PIM3 Q86V86 2/20 0.44
PIM2 Q9P1W9 2/20 0.44
GAK O14976 1/20 0.44
STK10 O94804 1/20 0.44
YES1 P07947 1/20 0.44
RET P07949 1/20 0.44
PDGFRB P09619 1/20 0.44
CSNK2A2 P19784 1/20 0.44
ACVR1 Q04771 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625776 0.89 PIM1 (0.55) PIM1FLT3KCNH2PIM3PIM2
SCHEMBL623999 0.85 MAPT (0.55) MAPTTP53
SCHEMBL624449 0.83 PIM1 (0.69) PIM1KCNH2PIM2DYRK1A
SCHEMBL624633 0.80 PIK3CA (0.47) ALDH1A1KDM4EMAPTHSD17B10HPGD
SCHEMBL624016 0.80 PIM1 (0.49) PIM1FLT3KCNH2PIM3PIM2
SCHEMBL623131 0.79 PIM1 (0.61) PIM1FLT3KCNH2PIM3PIM2
SCHEMBL628099 0.77 ALDH1A1 (0.49) ALDH1A1KDM4EMAPTHSD17B10HPGD
SCHEMBL624481 0.77 PIM1 (0.56) PIM1FLT3KCNH2PIM3PIM2
SCHEMBL623866 0.74 DYRK1A (0.48) PIM1KCNH2DYRK1A
SCHEMBL625034 0.74 PIM1 (0.54) PIM1FLT3KCNH2PIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed