SCHEMBL6248564

SCHEMBL6248564

NC(=O)C(=Cc1ccc2c(c1)CCO2)C(=O)N(c1cccc(C(F)(F)F)c1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
DYRK1A Q13627 3/20 0.38
DYRK1B Q9Y463 3/20 0.38
DYRK2 Q92630 2/20 0.38
RORC P51449 1/20 0.38
KCNH2 Q12809 2/20 0.38
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
FABP3 P05413 1/20 0.36
FABP4 P15090 1/20 0.36
GSK3B P49841 1/20 0.36
HSD11B1 P28845 1/20 0.36
RXFP1 Q9HBX9 2/20 0.35
DYRK3 O43781 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
NQO2 P16083 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CLK1 P49759 1/20 0.34
PIK3CA P42336 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6247880 0.80 RECQL (0.43) MAPTRECQLPKM
SCHEMBL6246748 0.77 GRK2 (0.40) MAPTRORCRXFP1RECQLPKM
SCHEMBL5145871 0.77 MAPT (0.60) MAPTRXFP1TP53POLBNPSR1
SCHEMBL6246353 0.76 RORC (0.40) RORCRXFP1RECQL
SCHEMBL6248753 0.76 EPHX1 (0.37) MAPTNQO2NPSR1RECQL
SCHEMBL6265380 0.76 LMNA (0.41) MAPTTP53POLB
SCHEMBL6248097 0.74 PTGS1 (0.44) MAPTRXFP1POLBNQO2NPSR1
SCHEMBL6247079 0.74 JAK2 (0.38) MAPTRORCRECQLPKM
SCHEMBL6248665 0.74 EPHX2 (0.47) MAPTRECQLPKMPKLR
SCHEMBL6246114 0.74 ALDH1A1 (0.48) MAPTPOLBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037196-A2 SUBSTITUTED 2-ARYLMETHYLENE-N-ARYL-N'-ARYL-MALONAMIDES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS CYTOVIA, INC. (US) 2005-04-28 WO disclosed