SCHEMBL6249306

SCHEMBL6249306

OCc1ccncc1CO

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AOC1 P19801 7/20 0.43
AOC3 Q16853 7/20 0.43
LOXL2 Q9Y4K0 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
HASPIN Q8TF76 1/20 0.41
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
RPS6KA3 P51812 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
ALOX12 P18054 1/20 0.36
CYP2A6 P11509 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29900474 1.00 AOC1 (0.43) AOC1AOC3LOXL2CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL31303524 0.97 AOC1 (0.45) AOC1AOC3LOXL2CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL21618217 0.97 AOC1 (0.45) AOC1AOC3LOXL2CYP11B1CYP11B2
SCHEMBL844847 0.86 CYP2E1 (0.43) AOC1AOC3LOXL2CYP11B1CYP11B2
SCHEMBL21352027 0.86 AOC1 (0.38) AOC1AOC3LOXL2CYP11B1CYP11B2
SCHEMBL5106244 0.86 CYP2E1 (0.43) AOC1AOC3LOXL2CYP11B1CYP11B2
SCHEMBL2642640 0.86 AOC1 (0.57) AOC1AOC3LOXL2CYP11B1CYP11B2
SCHEMBL2642637 0.86 AOC3 (0.41) AOC1AOC3LOXL2CYP11B1CYP11B2
SCHEMBL5109069 0.83 CYP2E1 (0.46) AOC1AOC3LOXL2CYP11B1CYP11B2
SCHEMBL5110078 0.83 CYP2E1 (0.46) AOC1AOC3LOXL2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240262792-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. 2024-08-08 US disclosed
US-20240245693-A1 COMPOSITIONS AND METHODS OF TISSUE REGENERATION THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-07-25 US disclosed
EP-4340940-A1 COMPOSITIONS AND METHODS OF TISSUE REGENERATION THERAPY The Regents of University of California (US) 2024-03-27 EP disclosed
US-11845724-B2 USP30 inhibitors and uses thereof VINCERE BIOSCIENCES, INC. (US) 2023-12-19 US disclosed
US-20230067476-A1 3-(5-HYDROXY-1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2023-03-02 US disclosed
US-20220315531-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. 2022-10-06 US disclosed
EP-4028385-A1 USP30 INHIBITORS AND USES THEREOF Vincere Biosciences, Inc. (US) 2022-07-20 EP disclosed
US-11192877-B2 3-(5-hydroxy-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2021-12-07 US disclosed
US-11186564-B2 Dual NAV1.2/5HT2a inhibitors for treating CNS disorders SUNOVION PHARMACEUTICALS INC. (US) 2021-11-30 US disclosed
WO-2021050992-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. (US) 2021-03-18 WO disclosed
WO-2021050992-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. (US) 2021-03-18 WO disclosed
US-20190194163-A1 DUAL NAV1.2/5HT2a INHIBITORS FOR TREATING CNS DISORDERS SUNOVION PHARMACEUTICALS INC. (US) 2019-06-27 US disclosed
WO-2018026371-A1 DUAL NAV1.2/5HT2A INHIBITORS FOR TREATING CNS DISORDERS SUNOVION PHARMACEUTICALS INC. (US) 2018-02-08 WO disclosed
WO-2005056013-A1 DPP-IV INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) GMBH (CH) 2005-06-23 WO disclosed
WO-2005056013-A1 DPP-IV INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) GMBH (CH) 2005-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190194163-A1 DUAL NAV1.2/5HT2a INHIBITORS FOR TREATING CNS DISORDERS SCN2A, HTR2A, HTR2C AOC1 4469/4885AOC3 2813/4885LOXL2 3303/4885
US-11186564-B2 Dual NAV1.2/5HT2a inhibitors for treating CNS disorders SCN2A, HTR2A, HTR2C AOC1 4469/4885AOC3 2813/4885LOXL2 3303/4885
US-11192877-B2 3-(5-hydroxy-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof XDH, HTR1D, RXFP1 AOC1 1589/4885AOC3 954/4885LOXL2 1042/4885
US-20230067476-A1 3-(5-HYDROXY-1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF XDH, HTR1D, RXFP1 AOC1 1589/4885AOC3 954/4885LOXL2 1042/4885
US-11845724-B2 USP30 inhibitors and uses thereof USP30, USP28, USP1 AOC1 3797/4885AOC3 3183/4885LOXL2 1859/4885
US-20220315531-A1 USP30 INHIBITORS AND USES THEREOF USP30, USP28, USP1 AOC1 3797/4885AOC3 3183/4885LOXL2 1859/4885
US-20240262792-A1 USP30 INHIBITORS AND USES THEREOF USP30, USP28, USP1 AOC1 3797/4885AOC3 3183/4885LOXL2 1859/4885
US-20240245693-A1 COMPOSITIONS AND METHODS OF TISSUE REGENERATION THERAPY ADORA2B, ADORA2A, ANXA3 AOC1 901/4885AOC3 463/4885LOXL2 2093/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.