SCHEMBL626165

SCHEMBL626165

CS(=O)(=O)N1CCC(Nc2nn3cc(-c4cncc(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.47
CDK2 P24941 11/20 0.42
CCNE1 P24864 10/20 0.42
F2RL3 Q96RI0 3/20 0.40
CDK1 P06493 7/20 0.38
CCNB1 P14635 7/20 0.38
CCND1 P24385 6/20 0.38
CDK6 Q00534 6/20 0.38
CDK4 P11802 5/20 0.38
CCND3 P30281 5/20 0.38
EPHX2 P34913 1/20 0.38
IDH1 O75874 1/20 0.38
IDH2 P48735 1/20 0.38
CCNB2 O95067 1/20 0.37
CCNE2 O96020 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
TNF P01375 1/20 0.36
TDO2 P48775 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626172 0.87 DYRK1A (0.38) IDO1CDK2CCNE1CDK1CCNB1
SCHEMBL624431 0.85 FYN (0.48) CDK2CCNE1F2RL3CDK1CCNB1
SCHEMBL626207 0.84 MAP3K12 (0.46) IDO1CDK2CCNE1CDK1CCNB1
SCHEMBL626187 0.84 JAK3 (0.38) IDO1CDK2CCNE1F2RL3CDK1
SCHEMBL626164 0.82 FYN (0.51) IDO1CDK2CCNE1CCND1CDK6
SCHEMBL626704 0.81 CCNE1 (0.43) IDO1CDK2CCNE1CDK1CCNB1
SCHEMBL624394 0.80 CCNE1 (0.41) IDO1CDK2CCNE1CDK1CCNB1
SCHEMBL623928 0.77 FYN (0.49) CDK2F2RL3CDK1CCND1CDK6
SCHEMBL625861 0.77 GPR119 (0.46) CDK2CCNE1CDK1CCNB1CCND1
SCHEMBL627168 0.75 CCNE1 (0.39) IDO1CDK2CCNE1CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed