SCHEMBL6265295

SCHEMBL6265295

NC(=O)/C(=C/c1ccc(C(F)(F)F)nc1)C(=O)N(c1cccc(C(F)(F)F)c1)c1ccc2ncccc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.38
CYP3A4 P08684 3/20 0.33
TSHR P16473 2/20 0.33
HSD17B10 Q99714 2/20 0.33
MTOR P42345 1/20 0.33
MDM2 Q00987 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CNR2 P34972 2/20 0.32
P4HB P07237 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
PARP1 P09874 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
KMT2A Q03164 2/20 0.32
TRPV1 Q8NER1 1/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
DOT1L Q8TEK3 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6248700 0.84 KMT2A (0.36) TSHRHSD17B10ALDH1A1P4HBKMT2A
SCHEMBL6292971 0.77 KDM4E (0.43) HSD17B10ALDH1A1CYP1A2KMT2A
SCHEMBL5144541 0.76 BRAF (0.49) BRAFCYP3A4TSHRHSD17B10ALDH1A1
SCHEMBL5144544 0.76 BRAF (0.49) BRAFCYP3A4TSHRHSD17B10ALDH1A1
SCHEMBL6246748 0.76 GRK2 (0.40) BRAFCYP3A4ALDH1A1CYP1A2P4HB
SCHEMBL6247880 0.75 RECQL (0.43) ALDH1A1P4HBKMT2AMEN1
SCHEMBL6246114 0.73 ALDH1A1 (0.48) ALDH1A1KMT2AMEN1POLBNPSR1
SCHEMBL6246207 0.73 LMNA (0.34) ALDH1A1CNR2KMT2AMEN1
SCHEMBL6246353 0.72 RORC (0.40) CYP3A4
SCHEMBL6248753 0.72 EPHX1 (0.37) ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037196-A2 SUBSTITUTED 2-ARYLMETHYLENE-N-ARYL-N'-ARYL-MALONAMIDES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS CYTOVIA, INC. (US) 2005-04-28 WO disclosed