SCHEMBL6265489

SCHEMBL6265489

O=C(O)c1ccc(OCC2CCN(c3ccc(Cl)cc3)C2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.58
ALDH1A1 P00352 3/20 0.53
MAPT P10636 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
LMNA P02545 1/20 0.53
MAPK1 P28482 1/20 0.53
HTT P42858 1/20 0.53
NOTUM Q6P988 1/20 0.50
HRH1 P35367 1/20 0.49
CCR3 P51677 1/20 0.49
KCNH2 Q12809 1/20 0.49
FFAR1 O14842 1/20 0.49
NR4A2 P43354 1/20 0.48
USP2 O75604 1/20 0.46
RBP4 P02753 1/20 0.45
TTR P02766 1/20 0.45
ACACB O00763 1/20 0.45
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6272089 0.97 ENPP2 (0.55) ENPP2ALDH1A1MAPTMEN1KMT2A
Hydrochloric Acid SCHEMBL9032597 0.96 ENPP2 (0.54) ENPP2ALDH1A1MAPTMEN1KMT2A
SCHEMBL6266696 0.93 ENPP2 (0.56) ENPP2ALDH1A1MAPTMEN1KMT2A
SCHEMBL6273298 0.88 MAPT (0.56) ENPP2ALDH1A1MAPTMEN1KMT2A
SCHEMBL8150260 0.88 RXRA (0.48) ENPP2ALDH1A1MAPTHRH1CCR3
SCHEMBL6270048 0.85 MAPT (0.53) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL6272036 0.85 NR4A2 (0.51) ALDH1A1MAPTLMNAHTTFFAR1
SCHEMBL6272295 0.82 NR4A2 (0.48) ALDH1A1MAPTLMNAHTTFFAR1
SCHEMBL6265368 0.82 DRD2 (0.50) ENPP2ALDH1A1MAPTMEN1KMT2A
Hydrochloric Acid SCHEMBL9032792 0.81 DRD2 (0.49) ENPP2ALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000620-B1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBITORS TAIHO PHARMACEUTICAL CO LTD (JP) 2005-12-07 EP disclosed
US-6166036-A Lp(a)-lowering agent and apolipoprotein (a) formation suppressing agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2000-12-26 US disclosed
EP-1000620-A1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBTORS TAIHO PHARMACEUTICAL COMPANY, LIMITED (JP) 2000-05-17 EP disclosed
EP-0393607-B1 Phenylcarboxylic acid derivatives having a hetero ring OTSUKA PHARMA CO LTD (JP) 1996-02-21 EP disclosed
US-5145865-A Fatty acid, cholesterol synthesis inhibitors; enzyme inhibitors; antilipemic agents OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1992-09-08 US disclosed