SCHEMBL6272089

SCHEMBL6272089

O=C(O)c1ccc(OCC2CCN(c3ccc(Oc4ccc(Cl)cc4)cc3)C2)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.55
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
MAPK1 P28482 1/20 0.50
HTT P42858 1/20 0.50
KMT2A Q03164 1/20 0.50
LTA4H P09960 9/20 0.48
NOTUM Q6P988 1/20 0.47
HRH1 P35367 1/20 0.47
CCR3 P51677 1/20 0.47
KCNH2 Q12809 1/20 0.47
FFAR1 O14842 2/20 0.47
NR4A2 P43354 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9032597 0.99 ENPP2 (0.54) ENPP2MEN1ALDH1A1LMNAMAPT
SCHEMBL6265489 0.97 ENPP2 (0.58) ENPP2MEN1ALDH1A1LMNAMAPT
SCHEMBL6266696 0.90 ENPP2 (0.56) ENPP2MEN1ALDH1A1LMNAMAPT
SCHEMBL6270048 0.89 MAPT (0.53) MEN1ALDH1A1LMNAMAPTMAPK1
SCHEMBL6272295 0.86 NR4A2 (0.48) ALDH1A1LMNAMAPTHTTFFAR1
SCHEMBL6273298 0.85 MAPT (0.56) ENPP2MEN1ALDH1A1LMNAMAPT
SCHEMBL8150260 0.85 RXRA (0.48) ENPP2ALDH1A1MAPTHRH1CCR3
SCHEMBL6272036 0.82 NR4A2 (0.51) ALDH1A1LMNAMAPTHTTFFAR1
SCHEMBL6265368 0.79 DRD2 (0.50) ENPP2MEN1ALDH1A1LMNAMAPT
SCHEMBL6267129 0.79 LMNA (0.53) ENPP2MEN1ALDH1A1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000620-B1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBITORS TAIHO PHARMACEUTICAL CO LTD (JP) 2005-12-07 EP disclosed
US-6166036-A Lp(a)-lowering agent and apolipoprotein (a) formation suppressing agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2000-12-26 US disclosed
EP-1000620-A1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBTORS TAIHO PHARMACEUTICAL COMPANY, LIMITED (JP) 2000-05-17 EP disclosed
EP-0393607-B1 Phenylcarboxylic acid derivatives having a hetero ring OTSUKA PHARMA CO LTD (JP) 1996-02-21 EP disclosed
US-5145865-A Fatty acid, cholesterol synthesis inhibitors; enzyme inhibitors; antilipemic agents OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1992-09-08 US disclosed