SCHEMBL6266142

SCHEMBL6266142

CC(C)(C)OC(=O)N1CCN(c2ccccc2-c2ccc(C=O)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 1/20 0.49
SMARCA4 P51532 1/20 0.49
PBRM1 Q86U86 1/20 0.49
CKS1B P61024 2/20 0.47
SKP1 P63208 2/20 0.47
SKP2 Q13309 2/20 0.47
BACE1 P56817 5/20 0.46
PDK2 Q15119 1/20 0.46
GPR119 Q8TDV5 3/20 0.45
AKT1 P31749 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
NAMPT P43490 1/20 0.43
KIT P10721 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20818663 0.87 CKS1B (0.58) SMARCA2SMARCA4PBRM1CKS1BSKP1
SCHEMBL29707355 0.86 CKS1B (0.50) SMARCA2SMARCA4PBRM1CKS1BSKP1
SCHEMBL6253535 0.84 GPR119 (0.53) SMARCA2SMARCA4PBRM1CKS1BSKP1
SCHEMBL209802 0.81 MAPT (0.64) PDK2GPR119ALDH1A1LMNAMAPT
SCHEMBL114482 0.80 GPR119 (0.53) SMARCA2SMARCA4PBRM1CKS1BSKP1
SCHEMBL22579225 0.80 MAPT (0.51) PDK2GPR119ALDH1A1LMNAMAPT
SCHEMBL12595780 0.79 ALDH1A1 (0.59) SMARCA2SMARCA4PBRM1GPR119ALDH1A1
SCHEMBL30479010 0.78 ALDH1A1 (0.58) SMARCA2SMARCA4PBRM1PDK2GPR119
SCHEMBL355504 0.78 ALDH1A1 (0.58) SMARCA2SMARCA4PBRM1PDK2GPR119
SCHEMBL6228319 0.78 GPR119 (0.49) SMARCA2SMARCA4PBRM1CKS1BSKP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592772-A2 5HT7 ANTAGONISTS AND INVERSE AGONISTS Pfizer Products Incorporated (US) 2005-11-09 EP disclosed
US-20040229874-A1 5HT7 Antagonists and inverse agonists PFIZER INC. 2004-11-18 US disclosed
WO-2004067703-A2 5HT7 ANTAGONISTS AND INVERSE AGONISTS PFIZER PRODUCTS INC. (US) 2004-08-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229874-A1 5HT7 Antagonists and inverse agonists HTR7, HTR1A, HTR1B SMARCA2 4569/4885SMARCA4 4431/4885PBRM1 3895/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.