SCHEMBL626698

SCHEMBL626698

COc1cncc(-c2cn3nc(N4CCCC4=O)sc3n2)c1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.52
CYP11B1 P15538 5/20 0.52
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAPT P10636 11/20 0.40
F2RL3 Q96RI0 1/20 0.40
THRB P10828 3/20 0.40
RXFP1 Q9HBX9 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626697 0.82 CYP11B2 (0.53) CYP11B2CYP11B1CYP1A2CYP3A4CYP2C9
SCHEMBL624950 0.77 MAPT (0.56) MAPTTHRBRXFP1
SCHEMBL625664 0.76 MAPT (0.58) MAPTTHRBRXFP1TP53
SCHEMBL627767 0.72 L3MBTL1 (0.44) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL1944169 0.71 FYN (0.53) MAPTF2RL3THRBRXFP1CA12
SCHEMBL532335 0.69 CA12 (0.53) CYP1A2CYP3A4CYP2C9CYP2C19F2RL3
SCHEMBL1945185 0.69 FYN (0.58) MAPTF2RL3THRBCA12CA1
SCHEMBL1762361 0.69 CYP11B1 (1.00) CYP11B2CYP11B1CYP1A2CYP3A4CYP2C9
SCHEMBL1945374 0.68 FYN (0.64) MAPTF2RL3CA12CA1CA2
SCHEMBL624431 0.68 FYN (0.48) MAPTF2RL3THRBCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed