SCHEMBL6271133

SCHEMBL6271133

Cn1c(CN2CCOCC2)ccc1C1CCCC[N]1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HRH3 Q9Y5N1 5/20 0.34
CYP2A13 Q16696 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6272806 0.96 CXCR4 (0.36) CXCR4KDM4EHRH3CYP2A13SMN1; SMN2
SCHEMBL5163035 0.79 CCR3 (0.50) KDM4ESIGMAR1ALDH1A1
SCHEMBL6273564 0.78 HRH3 (0.34) KDM4EHRH3SMN1; SMN2NPC1RAB9A
SCHEMBL5177492 0.78 ALDH1A1 (0.43) CXCR4KDM4EHRH3SMN1; SMN2KMT2A
SCHEMBL5175965 0.75 ALDH1A1 (0.43) CXCR4KDM4EHRH3SMN1; SMN2KMT2A
SCHEMBL4657761 0.74 HRH3 (0.52) CXCR4KDM4EHRH3CYP2A13SMN1; SMN2
SCHEMBL22561509 0.69 CYP2A13 (0.49) CXCR4KDM4EHRH3CYP2A13SMN1; SMN2
SCHEMBL2978126 0.67 GAA (0.41) HRH3SMN1; SMN2RAB9ATSHRALDH1A1
SCHEMBL4658989 0.66 DRD2 (0.54) KMT2ACYP3A4CYP2C19TSHRSIGMAR1
SCHEMBL2980038 0.66 GAA (0.42) HRH3SMN1; SMN2RAB9ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578416-A1 MEDICAMENTS CONTAINING SUBSTITUTED 2,5-DIAMINOMETHYL-1H-PYRROLES Grünenthal GmbH (DE) 2005-09-28 EP claimed
WO-2004058248-A1 MEDICAMENTS CONTAINING SUBSTITUTED 2,5-DIAMINOMETHYL-1H-PYRROLES Grünenthal GmbH (DE) 2004-07-15 WO claimed