SCHEMBL627210

SCHEMBL627210

Ic1cn2nc(N3CCCC4(CCCN4)CC3)sc2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.35
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
CHRND Q07001 1/20 0.34
CDC42BPB Q9Y5S2 12/20 0.33
ROCK1 Q13464 10/20 0.33
HRH4 Q9H3N8 1/20 0.33
CHEK1 O14757 1/20 0.33
AURKA O14965 1/20 0.33
RPS6KA5 O75582 1/20 0.33
CHEK2 O96017 1/20 0.33
MAPK3 P27361 1/20 0.33
MAPK1 P28482 1/20 0.33
AKT1 P31749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627209 0.78 HASPIN (0.40) PIM1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL627088 0.73 MAPT (0.32) MAPTTHRB
SCHEMBL627773 0.68 MAPT (0.43) MAPTTHRB
SCHEMBL627055 0.64 MAPT (0.48) MAPTTHRB
SCHEMBL38663548 0.59 CHRNB2 (0.57) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL1556564 0.57 CDC42BPB (0.54) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL24273708 0.57 CHRNA1 (0.36) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL4504835 0.56 NPC1 (0.54) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL21287570 0.55 PTPN11 (0.57) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL627245 0.55 F2RL3 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed