SCHEMBL627055

SCHEMBL627055

COC(=O)C1CCN(c2nn3cc(I)nc3s2)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPT P10636 15/20 0.48
THRB P10828 3/20 0.46
RXFP1 Q9HBX9 1/20 0.44
GAA P10253 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL628000 0.81 MAPT (0.42) MAPTTHRBRXFP1GAALMNA
SCHEMBL625664 0.76 MAPT (0.58) MAPTTHRBRXFP1
SCHEMBL627054 0.76 KDM4E (0.48) MAPTTHRBRXFP1KDM4ELMNA
SCHEMBL628100 0.76 MAPT (0.54) MAPTTHRBGAAKDM4ELMNA
SCHEMBL626106 0.73 THRB (0.49) MAPTTHRBRXFP1GAA
SCHEMBL628264 0.71 BTK (0.51) MAPTTHRB
SCHEMBL21724996 0.69 SMN1; SMN2 (0.49) MAPTKDM4ELMNAMEN1KMT2A
SCHEMBL15164461 0.69 SMN1; SMN2 (0.47) MAPTKDM4ELMNAMEN1KMT2A
SCHEMBL627088 0.68 MAPT (0.32) MAPTTHRB
SCHEMBL1700325 0.68 HPGD (0.62) MAPTKDM4ELMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed