SCHEMBL6286862

SCHEMBL6286862

CC(C(=O)NS(=O)(=O)CCNC(=O)OCc1ccccc1)c1ccccc1C(=O)c1ccsc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.39
CA1 P00915 3/20 0.39
ACHE P22303 2/20 0.39
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MMP2 P08253 3/20 0.38
MMP9 P14780 3/20 0.38
MMP3 P08254 2/20 0.38
MMP14 P50281 2/20 0.38
MMP1 P03956 1/20 0.38
MMP7 P09237 1/20 0.38
HTT P42858 1/20 0.37
SLC1A3 P43003 1/20 0.37
SLC1A1 P43005 1/20 0.37
KCNA5 P22460 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
CA5A P35218 1/20 0.35
MAPT P10636 1/20 0.35
KAT2B Q92831 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7116994 0.88 LMNA (0.39) CA2CA1ACHELMNAL3MBTL1
SCHEMBL6284179 0.80 C5AR1 (0.39) CA2CA1
SCHEMBL6285807 0.75 ADRA2C (0.47) CA2CA1ACHELMNASMN1; SMN2
SCHEMBL6332320 0.75 GLI1 (0.53) CA2CA1LMNASMN1; SMN2HTT
SCHEMBL6320504 0.73 CXCR1 (0.53) CA2CA1ACHELMNASMN1; SMN2
SCHEMBL6328423 0.71 GLI1 (0.52) CA2CA1ACHELMNASMN1; SMN2
SCHEMBL4420152 0.66 LMNA (0.58) CA2CA1LMNASMN1; SMN2HTT
SCHEMBL4409743 0.66 LMNA (0.58) CA2CA1LMNASMN1; SMN2HTT
SCHEMBL6283491 0.65 HTT (0.45) CA2CA1ACHELMNASMN1; SMN2
SCHEMBL4061201 0.65 LMNA (0.65) CA2CA1LMNASMN1; SMN2MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6887903-B1 N-(2-aryl-propionyl)-sulfonamides and pharmaceutical preparations containing them DOMPE S.P.A. (IT) 2005-05-03 US disclosed
US-6881755-B2 N-(2-aryl-propionyl)-sulfonamides and pharmaceutical preparations containing them Dompé S.p.A. (IT) 2005-04-19 US disclosed
US-20030216392-A1 N - ( 2 - aryl - propionyl ) - sulfonamides and pharmaceutical preparations containing them DOMPE S.P.A. 2003-11-20 US disclosed
EP-1123276-B1 N-(2-ARYL-PROPIONYL)-SULFONAMIDES AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM DOMPE SPA (IT) 2003-01-08 EP disclosed
EP-1123276-A1 N-(2-ARYL-PROPIONYL)-SULFONAMIDES AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM Dompe' S.P.A. (IT) 2001-08-16 EP disclosed
WO-2000024710-A1 N-(2-ARYL-PROPIONYL)-SULFONAMIDES AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM DOMPE' S.P.A. (IT) 2000-05-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030216392-A1 N - ( 2 - aryl - propionyl ) - sulfonamides and pharmaceutical preparations containing them ELANE, MPO, FPR1 CA2 2887/4885CA1 3899/4885ACHE 2071/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.