SCHEMBL6293045

SCHEMBL6293045

O=C1CSC(=O)N1c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.48
ALDH1A1 P00352 4/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KMT2A Q03164 8/20 0.47
MEN1 O00255 7/20 0.47
GAA P10253 5/20 0.46
POLB P06746 1/20 0.46
LMNA P02545 1/20 0.45
ELANE P08246 1/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPK1 P28482 1/20 0.44
RECQL P46063 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
EGFR P00533 1/20 0.41
KDR P35968 1/20 0.41
GFER P55789 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11689294 0.81 KMT2A (0.70) MGLLALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL12632654 0.81 F2 (0.52) MGLLALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL1421274 0.81 GAA (0.69) MGLLALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL181733 0.80 KMT2A (0.64) MGLLALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL3798127 0.78 KMT2A (0.52) MGLLALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL11025571 0.77 CA12 (0.61) ALDH1A1KMT2AMEN1GAAPOLB
SCHEMBL7297607 0.77 DHODH (0.51) ALDH1A1KMT2AMEN1GAAPOLB
SCHEMBL11028524 0.75 CA2 (0.43) ALDH1A1HPGDSMN1; SMN2KMT2AMEN1
SCHEMBL3780616 0.73 LMNA (0.67) MGLLALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL10570978 0.70 L3MBTL1 (0.44) MGLLALDH1A1SMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7939554-B2 Of Src homology protein tyrosine phosphatase 1; phenyl isothiazolones or a benzo-1,4-quinone; antineoplastic agents; immunostimulants inducing a cytokine response; side effect reduction THE CLEVELAND CLINIC FOUNDATION (US) 2011-05-10 US disclosed
US-20080103160-A1 Protein phosphatase inhibitors THE CLEVELAND CLINIC FOUNDATION 2008-05-01 US disclosed
US-20080051464-A1 Protein phosphatase inhibitors THE CLEVELAND CLINIC FOUNDATION 2008-02-28 US disclosed
WO-2008002641-A2 PROTEIN PHOSPHATASE INHIBITORS THE CLEVELAND CLINIC FOUNDATION (US) 2008-01-03 WO disclosed
US-6921760-B2 Aralkyl and aralkylidene heterocyclic lactams and imides PFIZER INC. (US) 2005-07-26 US disclosed
US-6627627-B2 Useful as psychotherapeutic agents PFIZER INC. 2003-09-30 US disclosed
EP-1339696-A1 BENZYL(IDENE)-LACTAMS AND THEIR USE AS 5HT1-RECEPTOR LIGANDS Pfizer Products Inc. (US) 2003-09-03 EP disclosed
EP-0929528-B1 ARALKYL AND ARALKYLIDENE HETEROCYCLIC LACTAMS AND IMIDES PFIZER (US) 2003-07-23 EP disclosed
US-6562813-B2 Psychological disorders; antiserotonin agents; headache therapy PFIZER INC. 2003-05-13 US disclosed
US-6472388-B2 PSYCHOTHERAPEUTIC AGENTS. PFIZER INC 2002-10-29 US disclosed
US-20020147194-A1 Aralkyl and aralkylidene heterocyclic lactams and imides PFIZER INC. 2002-10-10 US disclosed
US-6423708-B1 Aralkyl and aralkylidene heterocyclic lactams and imides PFIZER INC 2002-07-23 US disclosed
US-20020091117-A1 ARALKYL AND ARALKYLIDENE HETEROCYCLIC LACTAMS AND IMIDES PFIZER INC. 2002-07-11 US disclosed
US-20020091118-A1 ARALKYL AND ARALKYLIDENE HETEROCYCLIC LACTAMS AND IMIDES PFIZER INC. 2002-07-11 US disclosed
US-20020091119-A1 Aralkyl and aralkylidene heterocyclic lactams and imides PFIZER INC. 2002-07-11 US disclosed
WO-2002046167-A1 BENZYL (IDENE)-LACTAMS AND THEIR USE AS 5HT1-RECEPTOR LIGANDS PFIZER PRODUCTS INC. (US) 2002-06-13 WO disclosed
US-20020072519-A1 Aralkyl and aralkylidene heterocyclic lactams and imides PFIZER INC. 2002-06-13 US disclosed
US-6403592-B1 SEROTONIN REUPTAKE INHIBITORS PFIZER INC 2002-06-11 US disclosed
US-6380186-B1 PSYCHOTHERAPEUTIC AGENTS PFIZER INC 2002-04-30 US disclosed
US-20020049214-A1 Aralkyl and aralkylidene heterocyclic lactams and imides PFIZER PRODUCTS INC. 2002-04-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020091118-A1 ARALKYL AND ARALKYLIDENE HETEROCYCLIC LACTAMS AND IMIDES MRPL21, ARAF, ARL1 MGLL 368/4885ALDH1A1 1607/4885HPGD 1937/4885
US-20020091119-A1 Aralkyl and aralkylidene heterocyclic lactams and imides MRPL21, ARAF, ARL1 MGLL 368/4885ALDH1A1 1607/4885HPGD 1937/4885
US-20020147194-A1 Aralkyl and aralkylidene heterocyclic lactams and imides MRPL21, ARAF, ARL1 MGLL 368/4885ALDH1A1 1607/4885HPGD 1937/4885
US-20020049214-A1 Aralkyl and aralkylidene heterocyclic lactams and imides MRPL21, ARAF, ARL1 MGLL 284/4885ALDH1A1 1434/4885HPGD 2268/4885
US-20080103160-A1 Protein phosphatase inhibitors PPM1A, DUSP15, PPM1B MGLL 3271/4885ALDH1A1 1282/4885HPGD 1845/4885
US-20020072519-A1 Aralkyl and aralkylidene heterocyclic lactams and imides MRPL21, ARAF, ARL1 MGLL 368/4885ALDH1A1 1607/4885HPGD 1937/4885
US-20020091117-A1 ARALKYL AND ARALKYLIDENE HETEROCYCLIC LACTAMS AND IMIDES MRPL21, ARAF, ARL1 MGLL 368/4885ALDH1A1 1607/4885HPGD 1937/4885
US-20080051464-A1 Protein phosphatase inhibitors PPM1A, DUSP15, PPM1B MGLL 3271/4885ALDH1A1 1282/4885HPGD 1845/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.