SCHEMBL6295040

SCHEMBL6295040

CC(C)COc1ccc(-c2cc(NS(C)(=O)=O)ccc2Oc2ccc3cc(C#N)ccc3c2)c(C(=O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 11/20 0.43
SCN9A Q15858 2/20 0.40
PLA2G7 Q13093 2/20 0.37
NR3C1 P04150 3/20 0.36
PGR P06401 3/20 0.36
NR3C2 P08235 3/20 0.36
AR P10275 2/20 0.36
XDH P47989 1/20 0.35
SLC22A12 Q96S37 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7153794 0.95 BRD4 (0.40) BRD4SCN9APLA2G7NR3C1PGR
Trifluoroacetic Acid SCHEMBL7150674 0.84 PLA2G7 (0.37) BRD4SCN9APLA2G7SLC22A12
Trifluoroacetic Acid SCHEMBL7157237 0.84 PLA2G7 (0.39) SCN9APLA2G7SLC22A12
Trifluoroacetic Acid SCHEMBL7150670 0.83 PLA2G7 (0.41) SCN9APLA2G7SLC22A12
Trifluoroacetic Acid SCHEMBL7153144 0.79 BRD4 (0.43) BRD4SCN9APLA2G7PGRAR
SCHEMBL6295804 0.74 ALDH1A1 (0.40) SCN9AXDH
Trifluoroacetic Acid SCHEMBL6296006 0.74 BRD4 (0.43) BRD4SCN9APLA2G7
SCHEMBL6294972 0.73 PLAU (0.47) SCN9APLA2G7SLC22A12
SCHEMBL8506169 0.72 F3 (0.57)
SCHEMBL6300729 0.72 SLC22A12 (0.43) SCN9APLA2G7SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6916837-B2 Amidino derivatives and anticoagulants and thrombosis therapeutic agents containing them EISAI CO., LTD. (JP) 2005-07-12 US disclosed