SCHEMBL629939

SCHEMBL629939

CC(C)c1ccc(C[C@H](NC(=O)O[C@H]2CCCCN2S(=O)(=O)c2ccccc2)NC(=O)C(C)(C)CO)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 1/20 0.43
FKBP1A P62942 6/20 0.38
PKM P14618 1/20 0.37
ITGB1 P05556 2/20 0.37
ITGA5 P08648 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 1/20 0.37
BDKRB1 P46663 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
BCHE P06276 2/20 0.36
KCNQ1 P51787 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1381491 0.87 CCR4 (0.53) CCR4FKBP1APKMITGB1ITGA5
SCHEMBL630983 0.87 CCR4 (0.53) CCR4FKBP1APKMITGB1ITGA5
SCHEMBL630023 0.86 AKR1C3 (0.44) FKBP1APKMITGB1ITGA5ALDH1A1
SCHEMBL631075 0.80 FKBP1A (0.43) FKBP1APKMITGB1ITGA5TDP1
SCHEMBL630007 0.79 FKBP1A (0.48) FKBP1ATDP1LMNABDKRB1KCNQ1
SCHEMBL631251 0.78 ALDH1A1 (0.49) FKBP1APKMALDH1A1MAPK1NPSR1
SCHEMBL631233 0.78 FKBP1A (0.46) FKBP1APKMITGB1ITGA5ALDH1A1
SCHEMBL630767 0.76 ITGB1 (0.46) FKBP1APKMITGB1ITGA5ALDH1A1
SCHEMBL630470 0.76 MEN1 (0.48) FKBP1APKMITGB1ITGA5ALDH1A1
SCHEMBL631733 0.75 CCR4 (0.52) CCR4FKBP1APKMITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778637-B1 FKBP-binding composition and pharmaceutical use thereof AVENTIS PHARMA INC (US) 2012-02-22 EP claimed